SCHEMBL7013206

SCHEMBL7013206

Cc1cccc2nc(Cl)n(C)c(=O)c12

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.49
ELANE P08246 11/20 0.46
PARP1 P09874 2/20 0.46
CASR P41180 2/20 0.45
PIK3CD O00329 1/20 0.44
CTRB1 P17538 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7014708 0.83 ELANE (0.49) ELANEPARP1CASRPIK3CDCTRB1
SCHEMBL7011912 0.80 ELANE (0.46) ELANEPARP1CASRPIK3CDCTRB1
SCHEMBL2069228 0.80 ELANE (0.49) SMN1; SMN2ELANE
SCHEMBL10173803 0.80 PIK3CD (0.50) ELANEPARP1CASRPIK3CD
SCHEMBL16664255 0.78 PIK3CD (0.43) ELANEPARP1CASRPIK3CDCTRB1
SCHEMBL4402541 0.77 ESR2 (0.46) SMN1; SMN2ELANEPARP1PIK3CD
SCHEMBL1161604 0.76 PIK3CD (0.50) ELANEPARP1CASRPIK3CD
SCHEMBL28116231 0.75 PIK3CD (0.43) ELANEPARP1CASRPIK3CD
SCHEMBL2611507 0.74 KDM4E (0.64) SMN1; SMN2
SCHEMBL30879806 0.74 KDM4E (0.64) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed