SCHEMBL7013422

SCHEMBL7013422

CCOC(=O)C(C(=O)OCC)N1CCC(c2ccc3c(n2)NCCC3)CC1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 20/20 0.45
ITGB3 P05106 17/20 0.45
ITGB5 P18084 15/20 0.45
ITGB6 P18564 4/20 0.45
ITGB1 P05556 2/20 0.45
ITGA5 P08648 1/20 0.45
ITGB8 P26012 1/20 0.45
ITGA2B P08514 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7013425 0.95 ITGAV (0.47) ITGAVITGB3ITGB5ITGB6ITGB1
SCHEMBL8479505 0.84 ITGAV (0.49) ITGAVITGB3ITGB5ITGB6ITGB1
SCHEMBL8479508 0.80 ITGAV (0.49) ITGAVITGB3ITGB5ITGB6ITGB1
SCHEMBL8483637 0.78 ITGAV (0.47) ITGAVITGB3ITGB5ITGB6ITGB1
SCHEMBL2383101 0.77 ITGAV (0.44) ITGAVITGB3ITGB5ITGB6ITGB1
SCHEMBL7009416 0.77 ITGAV (0.41) ITGAVITGB3ITGB5ITGB6ITGB1
SCHEMBL13712259 0.75 ITGAV (0.53) ITGAVITGB3ITGB5ITGB6ITGB1
SCHEMBL2376065 0.75 ITGAV (0.49) ITGAVITGB6
SCHEMBL8483640 0.74 ITGAV (0.47) ITGAVITGB3ITGB5ITGB6ITGB1
SCHEMBL22893614 0.73 ITGAV (0.38) ITGAVITGB3ITGB5ITGB6ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946165-B1 INTEGRIN ANTAGONISTS MERCK & CO INC (US) 2003-04-09 EP disclosed
EP-0946165-A4 INTEGRIN ANTAGONISTS MERCK & CO INC (US) 2001-04-11 EP disclosed
EP-0946165-A1 INTEGRIN ANTAGONISTS Merck & Co., Inc. (US) 1999-10-06 EP disclosed
US-5952341-A VITRONECTIN RECEPTOR ANTAGONISTS FOR INHIBITING BONE RESORPTION, TREATING AND PREVENTING OSTEOPOROSIS, AND INHIBITING RESTENOSIS, DIABETIC RETINOPATHY, TUMOR, MACULAR DEGENERATION, ANGIOGENESIS, ATHEROSCLEROSIS, INFLAMMATION MERCK & CO., INC. (US) 1999-09-14 US disclosed
WO-1998018460-A1 INTEGRIN ANTAGONISTS MERCK & CO., INC. (US) 1998-05-07 WO disclosed