SCHEMBL7013452

SCHEMBL7013452

Cc1cccc(Sc2c(C)c[nH]c(=O)c2N)c1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.39
DAO P14920 2/20 0.39
NOTUM Q6P988 1/20 0.37
TYMS P04818 7/20 0.37
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35
HTR1A P08908 2/20 0.34
HTR3A P46098 2/20 0.34
XDH P47989 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MCL1 Q07820 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7011304 0.79 SMN1; SMN2 (0.44) IDO1DAONOTUMTYMSHTR1A
SCHEMBL9488631 0.70 AR (0.46) IDO1NOTUMHTR1AHTR3ASMN1; SMN2
SCHEMBL7013173 0.70 TYMS (0.32) IDO1DAOTYMSMCL1
SCHEMBL13915410 0.69 AR (0.45) IDO1NOTUMHTR1AHTR3ASMN1; SMN2
SCHEMBL29543680 0.68 ACHE (0.58) IDO1NOTUMDDB1CRBNHTR1A
SCHEMBL29468631 0.68 ACHE (0.58) IDO1NOTUMDDB1CRBNHTR1A
SCHEMBL575896 0.68 ACHE (0.58) IDO1NOTUMDDB1CRBNHTR1A
SCHEMBL11617247 0.68 IDO1 (0.50) IDO1DAONOTUMPRMT5WDR77
SCHEMBL10348868 0.67 ACHE (0.46) IDO1NOTUMDDB1CRBNHTR1A
SCHEMBL9488559 0.66 ACHE (0.41) IDO1NOTUMHTR1AHTR3ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0843663-B9 4-ARYL-THIO-PYRIDIN-2(1H)-ONES, DRUGS CONTAINING SAME, AND USES THEREOF FOR TREATING HIV-RELATED DISEASES CENTRE NAT RECH SCIENT (FR) 2003-10-29 EP disclosed
EP-0843663-B1 4-ARYL-THIO-PYRIDIN-2(1H)-ONES, DRUGS CONTAINING SAME, AND USES THEREOF FOR TREATING HIV-RELATED DISEASES CENTRE NAT RECH SCIENT (FR) 2003-04-09 EP disclosed
WO-1997005113-A1 4-ARYL-THIO-PYRIDIN-2(1H)-ONES, DRUGS CONTAINING SAME, AND USES THEREOF FOR TREATING HIV-RELATED DISEASES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 1997-02-13 WO disclosed