SCHEMBL7013500

SCHEMBL7013500

Cc1c(F)c(N)c(Cl)c2c1c(=O)c(C(=O)O)cn2-c1cc(N)c(F)cc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 5/20 0.40
ALDH1A1 P00352 2/20 0.39
HTT P42858 1/20 0.39
STAT3 P40763 1/20 0.39
TOP2A P11388 4/20 0.36
TOP2B Q02880 1/20 0.36
GSK3B P49841 1/20 0.36
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 2/20 0.35
KCNH2 Q12809 2/20 0.35
PIM1 P11309 2/20 0.35
HRH3 Q9Y5N1 1/20 0.35
POLB P06746 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HSP90AA1 P07900 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
CACNA1F O60840 1/20 0.33
MAPK1 P28482 1/20 0.33
CACNA1D Q01668 1/20 0.33
CACNA1S Q13698 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7005814 0.93 TOP1 (0.40) TOP1ALDH1A1HTTSTAT3TOP2A
SCHEMBL7008690 0.88 TOP1 (0.38) TOP1ALDH1A1HTTSTAT3TOP2A
SCHEMBL6576283 0.88 TOP1 (0.43) TOP1ALDH1A1HTTSTAT3TOP2A
SCHEMBL7006109 0.86 TOP1 (0.41) TOP1ALDH1A1HTTSTAT3TOP2A
SCHEMBL6581471 0.84 TOP2A (0.42) TOP1ALDH1A1HTTSTAT3TOP2A
SCHEMBL7009597 0.83 GSK3B (0.44) TOP1ALDH1A1HTTSTAT3TOP2A
SCHEMBL7011510 0.83 KCNH2 (0.41) TOP1ALDH1A1HTTSTAT3TOP2A
SCHEMBL7009868 0.82 TOP1 (0.39) TOP1ALDH1A1HTTSTAT3TOP2A
SCHEMBL7011082 0.81 STAT3 (0.43) TOP1ALDH1A1HTTSTAT3TOP2A
SCHEMBL6578587 0.81 TOP1 (0.54) TOP1ALDH1A1TOP2ATOP2BCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945435-B1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMA CO LTD (JP) 2003-08-13 EP disclosed
US-6136823-A BACTERICIDES OR VIRICIDES WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-0945435-A1 NOVEL PYRIDONECARBOXYLIC ACID DERIVATIVES OR SALTS THEREOF AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT WAKUNAGA PHARMACEUTICAL CO., LTD. (JP) 1999-09-29 EP disclosed