Bicarbonate

Bicarbonate

SCHEMBL7014228

O=C(O)O.O=C(c1ccc(F)cc1)N1CCSC1

nearest known ligand 0.53

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Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.53
ALDH1A1 P00352 2/20 0.53
HSD17B10 Q99714 1/20 0.53
DPP4 P27487 2/20 0.49
DPP7 Q9UHL4 1/20 0.49
HSD11B1 P28845 3/20 0.49
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48
CA14 Q9ULX7 1/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
ATM Q13315 1/20 0.47
SLC6A7 Q99884 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.46
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30566616 0.83 HPGD (0.56) HPGDALDH1A1HSD17B10DPP4MEN1
SCHEMBL3563805 0.80 HPGD (0.56) HPGDALDH1A1HSD17B10DPP4CA12
SCHEMBL94847 0.80 HPGD (0.56) HPGDALDH1A1HSD17B10DPP4
SCHEMBL22305103 0.77 CA12 (0.71) HPGDALDH1A1HSD11B1CA12CA1
SCHEMBL6985975 0.77 CA12 (0.71) HPGDALDH1A1HSD11B1CA12CA1
SCHEMBL23236678 0.76 ALDH1A1 (0.62) HPGDALDH1A1HSD17B10DPP4MEN1
SCHEMBL4669126 0.75 DPP4 (0.45) HPGDALDH1A1HSD17B10DPP4DPP7
SCHEMBL3047748 0.74 CA12 (0.63) ALDH1A1HSD11B1CA12CA1CA2
SCHEMBL31334408 0.73 HPGD (0.76) HPGDALDH1A1HSD11B1CA12CA1
SCHEMBL643480 0.73 ALDH1A1 (0.69) HPGDALDH1A1HSD11B1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1252163-B1 4-PYRIDYL-AND 2,4-PYRIMIDINYL-SUBSTITUTED PYRROLE DERIVATIVES AND THEIR USE IN PHARMACY MERCKLE GMBH (DE) 2003-09-24 EP disclosed
EP-1252163-A2 4-PYRIDYL-AND 2,4-PYRIMIDINYL-SUBSTITUTED PYRROLE DERIVATIVES AND THEIR USE IN PHARMACY MERCKLE GMBH (DE) 2002-10-30 EP disclosed
WO-2001057042-A2 4-PYRIDYL-AND 2,4-PYRIMIDINYL-SUBSTITUTED PYRROLE DERIVATIVES AND THEIR USE IN PHARMACY MERCKLE GMBH (DE) 2001-08-09 WO disclosed