SCHEMBL7014490

SCHEMBL7014490

C[C@H](Nc1nccc(Cl)n1)c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 4/20 0.59
LCK P06239 7/20 0.56
PLK1 P53350 1/20 0.52
JAK2 O60674 1/20 0.52
JAK3 P52333 1/20 0.52
ADRA1D P25100 1/20 0.51
HTR2C P28335 1/20 0.51
ADRA1A P35348 1/20 0.51
ADRA1B P35368 1/20 0.51
MAPK14 Q16539 4/20 0.51
IDH1 O75874 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27850412 0.87 IDH1 (0.51) HTR7LCKPLK1JAK2JAK3
SCHEMBL27850423 0.84 HTR7 (0.52) HTR7JAK2JAK3ADRA1DHTR2C
SCHEMBL4644412 0.83 HRH4 (0.49) HTR7LCK
SCHEMBL14629467 0.82 HTR7 (0.57) HTR7LCKPLK1JAK2JAK3
SCHEMBL7016449 0.81 IDH1 (0.55) HTR7ADRA1DADRA1AADRA1BIDH1
SCHEMBL28120957 0.81 HTR7 (0.57) HTR7LCKPLK1JAK2JAK3
SCHEMBL17076676 0.81 MAPK14 (0.56) HTR7LCKPLK1JAK2JAK3
SCHEMBL17076677 0.81 MAPK14 (0.56) HTR7LCKPLK1JAK2JAK3
SCHEMBL1600112 0.81 HTR7 (0.56) HTR7LCKPLK1JAK2JAK3
SCHEMBL10271508 0.78 HTR7 (0.56) HTR7LCKPLK1JAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1206265-B1 SRC KINASE INHIBITOR COMPOUNDS MERCK & CO INC (US) 2003-11-12 EP disclosed
US-6498165-B1 PYRIMIDINE COMPOUNDS; PROPHYLAXIS AND TREATMENT OF SUCH AS IMMUNE DISEASES, HYPERPROLIFERATIVE DISORDERS, CANCER, ANGIOGENSIS, ATHEROSCELEROSIS, GRAFT REJECTION, RHEUMATOID ARTHRITIS, PSORIASIS MERCK & CO., INC. 2002-12-24 US disclosed