SCHEMBL7014741

SCHEMBL7014741

Cn1c(S)nc2ccc(Cl)cc2c1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
RXFP1 Q9HBX9 3/20 0.49
KDM4E B2RXH2 3/20 0.48
HTT P42858 2/20 0.48
LMNA P02545 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
MAPT P10636 2/20 0.45
MAPK1 P28482 1/20 0.45
NPC1 O15118 2/20 0.44
HTR3A P46098 2/20 0.44
HRH4 Q9H3N8 2/20 0.44
HSD17B10 Q99714 1/20 0.43
CYP3A4 P08684 1/20 0.42
RAB9A P51151 1/20 0.42
ALDH1A1 P00352 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NLRP3 Q96P20 1/20 0.41
DPP4 P27487 1/20 0.41
HDAC3 O15379 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9919074 0.82 NPC1 (0.54) MEN1KMT2ARXFP1KDM4EHTT
SCHEMBL7010620 0.82 SMN1; SMN2 (0.49) MEN1KMT2AKDM4EHTTLMNA
SCHEMBL7018791 0.81 BACE1 (0.43) KDM4EHSD17B10
SCHEMBL15457139 0.78 KDM4E (0.50) MEN1KMT2ARXFP1KDM4EHTT
SCHEMBL3823391 0.78 MEN1 (0.47) MEN1KMT2ARXFP1KDM4EHTT
SCHEMBL3823961 0.77 MEN1 (0.46) MEN1KMT2ARXFP1KDM4EHTT
SCHEMBL31276870 0.77 KDM4E (0.70) MEN1KMT2ARXFP1KDM4EHTT
SCHEMBL9671456 0.77 KDM4E (0.51) MEN1KMT2AKDM4EHTTLMNA
SCHEMBL1161492 0.77 KDM4E (0.49) MEN1KMT2ARXFP1KDM4EHTT
SCHEMBL7012534 0.76 KDM4E (0.64) MEN1KMT2ARXFP1KDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed