SCHEMBL7015237

SCHEMBL7015237

Cc1cccc2nc(SCc3ccc(C(=O)c4ccc(Cl)cc4Cl)cc3)n(C)c(=O)c12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
THRB P10828 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
DRD2 P14416 5/20 0.42
TBXA2R P21731 5/20 0.42
TP53 P04637 2/20 0.42
MAPT P10636 2/20 0.42
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MAOA P21397 2/20 0.40
MAOB P27338 2/20 0.40
ALDH1A1 P00352 1/20 0.40
PKM P14618 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HDAC3 O15379 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7014463 0.90 MEN1 (0.49) MEN1KMT2ATDP1DRD2TBXA2R
SCHEMBL7018370 0.90 MEN1 (0.50) MEN1KMT2ATHRBTDP1DRD2
SCHEMBL7011506 0.87 MEN1 (0.55) MEN1KMT2ATDP1TP53MAPT
SCHEMBL7015464 0.86 KMT2A (0.60) MEN1KMT2ATDP1DRD2TBXA2R
SCHEMBL7018222 0.84 TDP1 (0.49) MEN1KMT2ATHRBTDP1DRD2
SCHEMBL7017095 0.84 MEN1 (0.45) MEN1KMT2ATHRBTDP1TP53
SCHEMBL7016710 0.84 MAOA (0.44) MEN1KMT2ATHRBTDP1TP53
SCHEMBL7017586 0.84 MEN1 (0.57) MEN1KMT2ATDP1TP53CYP1A2
SCHEMBL7101327 0.84 MEN1 (0.60) MEN1KMT2ATDP1TP53MAPT
SCHEMBL7015787 0.83 MEN1 (0.51) MEN1KMT2ATDP1TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed