SCHEMBL7015446

SCHEMBL7015446

COc1cc2nc(Cc3ccccc3)n(-c3ccc(C(O)(C(F)(F)F)C(F)(F)F)cc3)c(=O)c2c(Cl)c1OC

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
NPSR1 Q6W5P4 1/20 0.38
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
PGR P06401 3/20 0.36
RORA P35398 1/20 0.36
RORC P51449 1/20 0.36
RORB Q92753 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7021964 0.93 ALDH1A1 (0.48) ALDH1A1NPC1RAB9ANPSR1NR1H2
SCHEMBL7018132 0.92 ALDH1A1 (0.47) ALDH1A1NPC1RAB9ANPSR1NR1H2
SCHEMBL7016751 0.89 ALDH1A1 (0.48) ALDH1A1NPC1RAB9ANPSR1NR1H2
SCHEMBL7016130 0.87 ALDH1A1 (0.47) ALDH1A1NPC1RAB9ANPSR1NR1H2
SCHEMBL7022225 0.87 ALDH1A1 (0.48) ALDH1A1NPC1RAB9ANPSR1NR1H2
SCHEMBL7020884 0.85 ALDH1A1 (0.52) ALDH1A1NPC1RAB9ANPSR1CYP3A4
SCHEMBL7017347 0.85 ALDH1A1 (0.53) ALDH1A1NPC1RAB9ANPSR1PGR
SCHEMBL5062276 0.85 ALDH1A1 (0.55) ALDH1A1NPC1RAB9ANPSR1
SCHEMBL7020823 0.85 ALDH1A1 (0.43) ALDH1A1NPC1RAB9ANPSR1
SCHEMBL7018493 0.84 ALDH1A1 (0.45) ALDH1A1NPC1RAB9ANPSR1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003106435-A1 FUSED-RING PYRIMIDIN-4(3H)-ONE DERIVATIVES, PROCESSES FOR THE PREPARATION AND USES THEREOF SANKYO COMPANY, LIMITED (JP) 2003-12-24 WO claimed
WO-2003106435-A1 FUSED-RING PYRIMIDIN-4(3H)-ONE DERIVATIVES, PROCESSES FOR THE PREPARATION AND USES THEREOF SANKYO COMPANY, LIMITED (JP) 2003-12-24 WO disclosed