SCHEMBL7015648

SCHEMBL7015648

NC1CCN(c2c(F)cc3c(=O)n(OC(=O)C(F)(F)F)c(=O)n4c3c2SCC4)C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 2/20 0.40
GSK3A P49840 2/20 0.40
GSK3B P49841 2/20 0.40
PIM3 Q86V86 2/20 0.40
CSNK1G1 Q9HCP0 1/20 0.40
ALDH1A1 P00352 2/20 0.40
POLB P06746 1/20 0.40
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
TOP2A P11388 11/20 0.37
TOP2B Q02880 9/20 0.37
KDM4E B2RXH2 2/20 0.36
ADRA2B P18089 1/20 0.36
MAPK1 P28482 1/20 0.36
TOP1 P11387 4/20 0.36
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PRKD3 O94806 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7012922 0.89 KDM4E (0.36) ALDH1A1KDM4EADRA2BMAPK1HPGD
SCHEMBL6802345 0.82 PIM1 (0.43) PIM1GSK3AGSK3BPIM3CSNK1G1
SCHEMBL7011369 0.71 PRKD3 (0.43) PIM1GSK3AGSK3BPIM3ALDH1A1
SCHEMBL6807190 0.70 KDM4E (0.37) PIM1GSK3AGSK3BPIM3CSNK1G1
SCHEMBL6807192 0.70 KDM4E (0.37) PIM1GSK3AGSK3BPIM3CSNK1G1
SCHEMBL6800235 0.69 PIM1 (0.56) PIM1GSK3AGSK3BPIM3CSNK1G1
SCHEMBL7012086 0.69 KMT2A (0.43) PIM1GSK3AGSK3BPIM3CHRM2
SCHEMBL7013934 0.69 PRKD3 (0.39) PIM1GSK3AGSK3BPIM3ALDH1A1
SCHEMBL6803349 0.68 PIM1 (0.44) PIM1GSK3AGSK3BPIM3CSNK1G1
SCHEMBL7014855 0.67 TOP1 (0.42) PIM1GSK3AGSK3BPIM3POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1028950-B1 7-SUBSTITUTED QUINAZOLIN-2,4-DIONES USEFUL AS ANTIBACTERIAL AGENTS WARNER LAMBERT CO (US) 2003-05-02 EP claimed