SCHEMBL7016296

SCHEMBL7016296

CC(O)c1c(N(C)C)cnn(C(C)(C)C)c1=O

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.33
NPSR1 Q6W5P4 1/20 0.33
NPC1 O15118 2/20 0.32
LMNA P02545 2/20 0.32
RAB9A P51151 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
MEN1 O00255 1/20 0.30
GALR3 O60755 1/20 0.30
NR2F2 P24468 1/20 0.30
GPR183 P32249 1/20 0.30
KMT2A Q03164 1/20 0.30
GPR35 Q9HC97 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7011309 0.80 KAT2B (0.37) SMN1; SMN2NPC1LMNARAB9ACYP1A2
SCHEMBL7017794 0.74 NPC1 (0.33) SMN1; SMN2NPC1LMNARAB9ACYP1A2
SCHEMBL24498709 0.72 SMN1; SMN2 (0.39) SMN1; SMN2NPSR1NPC1LMNARAB9A
SCHEMBL7013194 0.72 LMNA (0.33) SMN1; SMN2NPC1LMNARAB9ACYP1A2
SCHEMBL17582551 0.65 PIK3CD (0.46) SMN1; SMN2NPC1LMNARAB9ACYP3A4
SCHEMBL8550187 0.64 TSHR (0.38) SMN1; SMN2NPSR1NPC1LMNARAB9A
SCHEMBL8542209 0.64 SMN1; SMN2 (0.38) SMN1; SMN2NPSR1NPC1LMNARAB9A
SCHEMBL14012593 0.62 TSHR (0.39) SMN1; SMN2NPSR1NPC1LMNARAB9A
SCHEMBL9237010 0.61 SMN1; SMN2 (0.38) SMN1; SMN2NPSR1NPC1LMNARAB9A
SCHEMBL12410744 0.60 TSHR (0.41) SMN1; SMN2NPSR1NPC1LMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed