SCHEMBL7016568

SCHEMBL7016568

CC(C)(CC(=O)O)Cc1ccc(OCCCNc2ccccn2)cc1C#N

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 18/20 0.48
ITGAV P06756 18/20 0.48
ITGB1 P05556 7/20 0.48
ITGB5 P18084 4/20 0.48
ITGB6 P18564 3/20 0.48
MDM4 O15151 1/20 0.45
MDM2 Q00987 1/20 0.45
ITGA2B P08514 4/20 0.45
ITGA5 P08648 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL6802228 0.97 ITGB3 (0.48) ITGB3ITGAVITGB1ITGB5ITGB6
SCHEMBL6804811 0.91 ITGB3 (0.48) ITGB3ITGAVITGB1ITGB5ITGB6
SCHEMBL6804856 0.90 ITGB3 (0.42) ITGB3ITGAVITGB1ITGB5ITGB6
SCHEMBL6809475 0.89 ITGB3 (0.49) ITGB3ITGAVITGB1ITGB5ITGB6
SCHEMBL7018419 0.88 ITGB3 (0.42) ITGB3ITGAVITGB1ITGB5ITGB6
Trifluoroacetic Acid SCHEMBL6806426 0.88 ITGB3 (0.48) ITGB3ITGAVITGB1ITGB5ITGB6
Trifluoroacetic Acid SCHEMBL6804895 0.86 ITGB3 (0.49) ITGB3ITGAVITGB1ITGB5ITGB6
SCHEMBL6804884 0.86 ITGB3 (0.51) ITGB3ITGAVITGB1ITGB5ITGB6
Trifluoroacetic Acid SCHEMBL6809448 0.83 ITGB3 (0.50) ITGB3ITGAVITGB1ITGB5ITGB6
SCHEMBL6805351 0.82 ITGB3 (0.46) ITGB3ITGAVITGB1ITGB5ITGB6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1313705-A1 GEM-SUBSTITUTED ALPHA V BETA 3 INTEGRIN ANTAGONISTS Pharmacia Corporation (US) 2003-05-28 EP claimed
US-6531494-B1 Gem-substituted αvβ3 antagonists PHARMACIA CORPORATION 2003-03-11 US claimed
WO-2002018340-A1 GEM-SUBSTITUTED α v β 3 INTEGRIN ANTAGONISTS PHARMACIA CORPORATION (US) 2002-03-07 WO claimed
EP-1313705-A1 GEM-SUBSTITUTED ALPHA V BETA 3 INTEGRIN ANTAGONISTS Pharmacia Corporation (US) 2003-05-28 EP disclosed
US-6531494-B1 Gem-substituted αvβ3 antagonists PHARMACIA CORPORATION 2003-03-11 US disclosed
WO-2002018340-A1 GEM-SUBSTITUTED α v β 3 INTEGRIN ANTAGONISTS PHARMACIA CORPORATION (US) 2002-03-07 WO disclosed