SCHEMBL7017444

SCHEMBL7017444

COc1cc2c(cc1C=O)C(C)C(=O)N2C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.46
KDM4E B2RXH2 1/20 0.46
TSHR P16473 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
MAPT P10636 2/20 0.46
BRD4 O60885 5/20 0.40
CCL2 P13500 1/20 0.40
GAA P10253 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
PRKDC P78527 1/20 0.36
ERN1 O75460 2/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MCOLN3 Q8TDD5 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
NPC1 O15118 1/20 0.33
POLB P06746 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27578391 0.77 ALDH1A1 (0.44) ALDH1A1KDM4ETSHRTDP1MAPT
SCHEMBL6074170 0.76 ALDH1A1 (0.43) ALDH1A1KDM4ETSHRTDP1MAPT
SCHEMBL5165016 0.76 ALDH1A1 (0.43) ALDH1A1KDM4ETSHRTDP1MAPT
SCHEMBL6073770 0.76 ALDH1A1 (0.43) ALDH1A1KDM4ETSHRTDP1MAPT
SCHEMBL4148886 0.76 ALDH1A1 (0.43) ALDH1A1KDM4ETSHRTDP1MAPT
SCHEMBL6604704 0.73 ALDH1A1 (0.49) ALDH1A1KDM4ETSHRTDP1MAPT
SCHEMBL6073885 0.73 ALDH1A1 (0.46) ALDH1A1KDM4ETSHRTDP1MAPT
SCHEMBL6608851 0.73 ALDH1A1 (0.46) ALDH1A1KDM4ETSHRTDP1MAPT
SCHEMBL8532730 0.72 BRD4 (0.52) ALDH1A1TSHRMAPTBRD4CCL2
SCHEMBL25295086 0.70 CYP2A6 (0.38) ALDH1A1KDM4ETSHRMAPTBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1272484-A2 BENZOAMIDE PIPERIDINE COMPOUNDS AS SUBSTANCE P ANTAGONISTS Pfizer Products Inc. (US) 2003-01-08 EP disclosed
WO-2001077100-A2 BENZOAMIDE PIPERIDINE COMPOUNDS AS SUBSTANCE P ANTAGONISTS PFIZER PRODUCTS INC. (US) 2001-10-18 WO disclosed