SCHEMBL7017695

SCHEMBL7017695

COc1cc2c(=O)n(-c3ccc(C(O)(C(F)(F)F)C(F)(F)F)cc3)c(Cc3ccccc3)nc2cc1O

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.53
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
NPSR1 Q6W5P4 1/20 0.43
KMT2A Q03164 2/20 0.42
PDE10A Q9Y233 2/20 0.42
CYP3A4 P08684 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
HIF1A Q16665 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7015149 0.96 ALDH1A1 (0.53) ALDH1A1NPC1RAB9ANPSR1KMT2A
SCHEMBL5062276 0.94 ALDH1A1 (0.55) ALDH1A1NPC1RAB9ANPSR1PDE10A
SCHEMBL7020461 0.92 ALDH1A1 (0.52) ALDH1A1NPC1RAB9ANPSR1KMT2A
SCHEMBL7020089 0.92 ALDH1A1 (0.52) ALDH1A1NPC1RAB9ANPSR1KMT2A
SCHEMBL7018345 0.91 ALDH1A1 (0.52) ALDH1A1NPC1RAB9ANPSR1KMT2A
SCHEMBL7015283 0.90 ALDH1A1 (0.52) ALDH1A1NPC1RAB9ANPSR1KMT2A
SCHEMBL7016929 0.90 ALDH1A1 (0.50) ALDH1A1NPC1RAB9ANPSR1PDE10A
SCHEMBL7025842 0.90 ALDH1A1 (0.50) ALDH1A1NPC1RAB9ANPSR1PDE10A
SCHEMBL7018834 0.90 ALDH1A1 (0.50) ALDH1A1NPC1RAB9ANPSR1PDE10A
SCHEMBL7019149 0.90 ALDH1A1 (0.50) ALDH1A1NPC1RAB9ANPSR1PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003106435-A1 FUSED-RING PYRIMIDIN-4(3H)-ONE DERIVATIVES, PROCESSES FOR THE PREPARATION AND USES THEREOF SANKYO COMPANY, LIMITED (JP) 2003-12-24 WO disclosed