SCHEMBL7017986

SCHEMBL7017986

C=C1C=C(c2ccccc2)C(c2ccccc2)=C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.44
BACE1 P56817 3/20 0.44
MAOA P21397 2/20 0.41
MAOB P27338 1/20 0.41
MAPK1 P28482 3/20 0.39
HSD17B10 Q99714 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
CYP3A4 P08684 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39
PTPN1 P18031 2/20 0.38
PTPRC P08575 1/20 0.38
PTPRF P10586 1/20 0.38
CDC25B P30305 1/20 0.38
HSD17B3 P37058 1/20 0.38
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
TDO2 P48775 1/20 0.33
POLB P06746 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
ADORA2A P29274 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1026969 0.73 ALDH1A1 (0.47) ALDH1A1BACE1MAOAMAOBMAPK1
SCHEMBL12480578 0.71 BACE1 (0.60) ALDH1A1BACE1MAOAMAOBPTPN1
SCHEMBL26135886 0.69 BACE1 (0.76) ALDH1A1BACE1MAOAMAOBMAPK1
Biphenyl SCHEMBL5586130 0.66 ALDH1A1 (0.82) ALDH1A1MAOAMAPK1HSD17B10TDP1
Biphenyl SCHEMBL388156 0.66 ALDH1A1 (0.82) ALDH1A1MAOAMAPK1HSD17B10TDP1
Biphenyl SCHEMBL5797043 0.65 ALDH1A1 (0.53) ALDH1A1MAOAMAPK1HSD17B10TDP1
Biphenyl SCHEMBL164 0.65 ALDH1A1 (1.00) ALDH1A1MAOAMAPK1HSD17B10TDP1
Biphenyl SCHEMBL1358618 0.65 ALDH1A1 (1.00) ALDH1A1MAOAMAPK1HSD17B10TDP1
SCHEMBL29560186 0.65 ALDH1A1 (1.00) ALDH1A1MAOAMAPK1HSD17B10TDP1
Biphenyl SCHEMBL2548048 0.65 ALDH1A1 (1.00) ALDH1A1MAOAMAPK1HSD17B10TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6214762-B1 REACTION OF METAL FULVENE COMPLEX AND UNSATURATED COMPOUND INSERTION COMPLEXES AND THE USE THEREOF AS CATALYSTS FOR THE POLYMERIZATION OF OLEFINS AND/OR DIENES AND AS HYDROGENATION CATALYSTS. BAYER AKTIENGESELLSCHAFT (DE) 2001-04-10 US claimed
EP-0980872-A2 Catalysts based upon fulvene-metal complexes Bayer Aktiengesellschaft (DE) 2000-02-23 EP claimed
EP-1185541-B1 CATALYST SYSTEM ON THE BASIS OF FULVENE COMPOUNDS BAYER AG (DE) 2003-01-15 EP disclosed
US-6403735-B1 REACTING TRANSITION METAL COMPOUND WITH FULVENE COMPOUND IN PRESENCE OF REDUCING AGENT BAYER AKTIENGESELLSCHAFT (DE) 2002-06-11 US disclosed
US-20020010084-A1 Method for producting fulvene metal complexes BECKE SIGURD (DE) 2002-01-24 US disclosed
US-6258744-B1 OLEFIN POLYMERIZATION CATALYST BAYER AKTIENGESELLSCHAFT (DE) 2001-07-10 US disclosed
US-6214762-B1 REACTION OF METAL FULVENE COMPLEX AND UNSATURATED COMPOUND INSERTION COMPLEXES AND THE USE THEREOF AS CATALYSTS FOR THE POLYMERIZATION OF OLEFINS AND/OR DIENES AND AS HYDROGENATION CATALYSTS. BAYER AKTIENGESELLSCHAFT (DE) 2001-04-10 US disclosed
EP-1028968-A1 METHOD FOR PRODUCING FULVENE METAL COMPLEXES BAYER AG (DE) 2000-08-23 EP disclosed
EP-0982319-A2 Catalyst system based on fulvene-cyclopentadienyl-metal complexes Bayer Aktiengesellschaft (DE) 2000-03-01 EP disclosed
EP-0980872-A2 Catalysts based upon fulvene-metal complexes Bayer Aktiengesellschaft (DE) 2000-02-23 EP disclosed
WO-1999024445-A1 METHOD FOR PRODUCING FULVENE METAL COMPLEXES BAYER AKTIENGESELLSCHAFT (DE) 1999-05-20 WO disclosed