Dimethylamine

Dimethylamine

SCHEMBL7018332

CNC.COC(=O)c1cccc(OC)c1S(=O)(=O)O

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.47
HSD17B10 Q99714 3/20 0.47
TSHR P16473 2/20 0.47
MAPT P10636 2/20 0.47
MAPK1 P28482 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA5A P35218 1/20 0.44
CA9 Q16790 1/20 0.44
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 3/20 0.44
POLB P06746 1/20 0.44
ATM Q13315 1/20 0.44
LMNA P02545 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
BACE1 P56817 1/20 0.43
SLC6A3 Q01959 1/20 0.43
CTSD P07339 1/20 0.41
CFTR P13569 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18762909 0.87 CA12 (0.42) GAAHSD17B10TSHRMAPTMAPK1
SCHEMBL433518 0.85 CA1 (0.53) HSD17B10TSHRMAPTL3MBTL1CA1
SCHEMBL3965219 0.83 CA1 (0.51) HSD17B10TSHRMAPTL3MBTL1CA1
SCHEMBL4178504 0.83 CA1 (0.51) HSD17B10TSHRMAPTL3MBTL1CA1
SCHEMBL375000 0.83 CA1 (0.51) HSD17B10TSHRMAPTL3MBTL1CA1
Water SCHEMBL27375204 0.83 CA1 (0.51) HSD17B10TSHRMAPTL3MBTL1CA1
SCHEMBL27647423 0.83 CA1 (0.51) HSD17B10TSHRMAPTL3MBTL1CA1
SCHEMBL7025204 0.83 HSD17B10 (0.48) GAAHSD17B10TSHRMAPTMAPK1
SCHEMBL7032454 0.83 CA1 (0.57) GAAHSD17B10TSHRMAPTMAPK1
SCHEMBL9815155 0.82 HTT (0.53) GAAHSD17B10TSHRMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0574174-B1 Angiotensin II antagonists LILLY CO ELI (US) 2003-08-13 EP disclosed
CN-1045768-C Angiotension II antagonists LILLY CO ELI (US) 1999-10-20 CN disclosed
US-5693633-A Angiotensin II antagonists ELI LILLY AND COMPANY (US) 1997-12-02 US disclosed
US-5612360-A AROMATIC N-HETEROCYCLIC COMPOUNDS AS HYPOTENSIVE AGENTS WITH ACID GROUPS, SULFONYLCARBOXAMIDES OR TETRAZOLE GROUPS ELI LILLY AND COMPANY (US) 1997-03-18 US disclosed
US-5569768-A USEFUL IN TREATING HYPERTENSION, CONGESTIVE HEART FAILURE, GLAUCOMA AND RENAL INSUFFICIENCY ELI LILLY AND COMPANY (US) 1996-10-29 US disclosed
US-5556981-A Angiotensin II antagonist intermediates ELI LILLY AND COMPANY (US) 1996-09-17 US disclosed
US-5484780-A CARDIOVASCULAR, HYPOTENSIVE ELI LILLY AND COMPANY (US) 1996-01-16 US disclosed
CN-1101908-A Angiotensin II antagonists LILLY CO ELI (US) 1995-04-26 CN disclosed
US-5401851-A Preparation of proline derivatives ELI LILLY AND COMPANY (US) 1995-03-28 US disclosed
CN-1085897-A Angiotension II antagonists LILLY CO ELI (US) 1994-04-27 CN disclosed
EP-0574174-A2 Angiotensin II antagonists ELI LILLY AND COMPANY (US) 1993-12-15 EP disclosed
EP-0573271-A1 Angiotensin II antagonists ELI LILLY AND COMPANY (US) 1993-12-08 EP disclosed