SCHEMBL7019199

SCHEMBL7019199

Cn1c(S)nc2cccc(C(=O)O)c2c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.44
ALDH1A1 P00352 2/20 0.41
HSD17B10 Q99714 2/20 0.40
KDM4E B2RXH2 3/20 0.40
CASP1 P29466 2/20 0.40
CASP7 P55210 2/20 0.40
CAMKK1 Q8N5S9 2/20 0.38
CAMKK2 Q96RR4 2/20 0.38
CSNK2A2 P19784 1/20 0.38
CSNK2B P67870 1/20 0.38
CSNK2A1 P68400 1/20 0.38
PIM3 Q86V86 1/20 0.38
DYRK2 Q92630 1/20 0.38
MKNK1 Q9BUB5 1/20 0.38
PIM2 Q9P1W9 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
MAPT P10636 2/20 0.37
ADORA2B P29275 1/20 0.37
CYP1A2 P05177 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7016252 0.76 ELANE (0.48) ALDH1A1HSD17B10KDM4ECASP1CASP7
SCHEMBL15840320 0.71 PARP1 (0.42) DHODHKDM4EKMT2A
SCHEMBL11247053 0.70 KDM4E (0.59) ALDH1A1HSD17B10KDM4ECASP1CASP7
SCHEMBL9532680 0.70 KDM4E (0.63) ALDH1A1HSD17B10KDM4EMAPTSMN1; SMN2
SCHEMBL29683984 0.66 ALDH1A1 (0.53) DHODHALDH1A1HSD17B10KDM4EMEN1
SCHEMBL28253069 0.65 DHODH (0.40) DHODHALDH1A1HSD17B10KDM4ECYP1A2
SCHEMBL10466519 0.64 ALDH1A1 (0.50) DHODHALDH1A1HSD17B10KDM4EDYRK2
SCHEMBL10465588 0.64 ALDH1A1 (0.46) DHODHALDH1A1HSD17B10KDM4ECASP7
SCHEMBL689778 0.63 HSD17B10 (0.64) ALDH1A1HSD17B10KDM4EMEN1KMT2A
SCHEMBL29404347 0.63 HSD17B10 (0.78) ALDH1A1HSD17B10KDM4ECASP7MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed