SCHEMBL7021080

SCHEMBL7021080

CN(C)CCOc1ccc(-n2cc(-c3ccccn3)cc(-c3ccccc3Cl)c2=O)cc1.O=c1c(-c2ccccc2Cl)cc(-c2ccccn2)cn1-c1ccc(O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 1/20 0.46
GRIA3 P42263 1/20 0.46
PDE4D Q08499 1/20 0.46
MCHR1 Q99705 1/20 0.43
ACVR1B P36896 1/20 0.41
TGFBR1 P36897 1/20 0.41
ESR1 P03372 10/20 0.40
KDR P35968 1/20 0.40
RIPK2 O43353 1/20 0.39
ACVR1 Q04771 1/20 0.39
NOD2 Q9HC29 1/20 0.39
ESRRG P62508 5/20 0.39
ESRRB O95718 4/20 0.39
ESR2 Q92731 3/20 0.39
FGFR1 P11362 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1882345 0.96 GRIA1 (0.50) GRIA1GRIA3PDE4DMCHR1ACVR1B
SCHEMBL1884211 0.92 GRIA1 (0.48) GRIA1GRIA3PDE4DMCHR1ACVR1B
SCHEMBL1881496 0.88 GRIA1 (0.49) GRIA1GRIA3PDE4DMCHR1ACVR1B
SCHEMBL6732337 0.87 GRIA1 (0.51) GRIA1GRIA3PDE4DESR1KDR
SCHEMBL1884441 0.87 GRIA1 (0.58) GRIA1GRIA3PDE4DESR1ESR2
SCHEMBL1884751 0.82 GRIA1 (0.53) GRIA1GRIA3PDE4DMCHR1ACVR1B
SCHEMBL1884295 0.82 GRIA1 (0.55) GRIA1GRIA3PDE4DTGFBR1KDR
SCHEMBL1882344 0.80 GRIA1 (0.49) GRIA1GRIA3PDE4DMCHR1RIPK2
SCHEMBL1891974 0.80 GRIA1 (0.47) GRIA1GRIA3PDE4DRIPK2ACVR1
SCHEMBL2961989 0.79 GRIA1 (0.68) GRIA1GRIA3PDE4DMCHR1ACVR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1300396-A1 1,2-DIHYDROPYRIDINE COMPOUNDS, PROCESS FOR PREPARATION OF THE SAME AND USE THEREOF Eisai Co., Ltd. (JP) 2003-04-09 EP disclosed