SCHEMBL7022406

SCHEMBL7022406

C#Cc1cccc(Nc2ncnc3c2ccn3C)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 14/20 0.57
GAK O14976 3/20 0.57
FBP1 P09467 2/20 0.57
ALDH1A1 P00352 1/20 0.57
MAPT P10636 1/20 0.57
ERBB2 P04626 3/20 0.54
ERBB4 Q15303 2/20 0.54
TP53 P04637 1/20 0.54
AURKA O14965 2/20 0.52
RPS6KB1 P23443 1/20 0.52
ABL1 P00519 2/20 0.52
BCR P11274 2/20 0.52
RIPK2 O43353 2/20 0.52
BUB1 O43683 2/20 0.52
STK10 O94804 2/20 0.52
MAP3K1 Q13233 2/20 0.52
PIP4K2C Q8TBX8 2/20 0.52
SLK Q9H2G2 2/20 0.52
KDR P35968 2/20 0.52
LMNA P02545 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7017577 0.99 EGFR (0.56) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL7022884 0.82 EGFR (0.60) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL29110509 0.81 EGFR (0.67) EGFRFBP1ERBB2AURKAAURKB
SCHEMBL4741962 0.81 EGFR (0.58) EGFRFBP1ALDH1A1MAPTERBB2
SCHEMBL13214883 0.80 ABL1 (0.65) EGFRALDH1A1MAPTERBB2ABL1
SCHEMBL7023791 0.80 EGFR (0.49) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL7018724 0.79 EGFR (0.59) EGFRGAKFBP1ALDH1A1MAPT
Hydrochloric Acid SCHEMBL7021265 0.79 FBP1 (0.48) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL7018558 0.78 KDR (0.48) EGFRGAKFBP1ALDH1A1MAPT
SCHEMBL29110515 0.78 EGFR (0.60) EGFRMAPTERBB2ERBB4TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0831829-B1 HETEROCYCLIC RING-FUSED PYRIMIDINE DERIVATIVES PFIZER (US) 2003-08-20 EP claimed
CN-1141298-A Pyrimidine-fused heterocyclic compound anti-cancer agents PFIZER (US) 1997-01-29 CN claimed
CN-1141298-A Pyrimidine-fused heterocyclic compound anti-cancer agents PFIZER (US) 1997-01-29 CN disclosed