SCHEMBL7023741

SCHEMBL7023741

O=c1[nH]c(=O)c2cc(CN3CCOCC3)ccc2[nH]1

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.62
TNKS O95271 1/20 0.49
JAK2 O60674 1/20 0.48
TYMP P19971 1/20 0.48
CHEK1 O14757 2/20 0.47
HSD17B10 Q99714 3/20 0.46
HRH3 Q9Y5N1 1/20 0.46
MAPT P10636 2/20 0.46
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 2/20 0.46
GAA P10253 1/20 0.46
ALOX15 P16050 1/20 0.46
HPGD P15428 1/20 0.45
CDK4 P11802 1/20 0.44
CCND1 P24385 1/20 0.44
CDK2 P24941 1/20 0.44
CDK7 P50613 1/20 0.44
NCF1 P14598 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18643633 0.76 PARP1 (0.56) PARP1TNKSHSD17B10HRH3KDM4E
SCHEMBL31061696 0.76 PARP1 (1.00) PARP1TNKSHSD17B10MAPTKDM4E
SCHEMBL7029687 0.76 PDE3A (0.55) HSD17B10MAPTKDM4EALDH1A1ALOX15
Hydrochloric Acid SCHEMBL6406540 0.75 PARP1 (0.97) PARP1TNKSHSD17B10MAPTKDM4E
SCHEMBL18643551 0.74 PARP1 (0.54) PARP1TNKSHSD17B10MAPTKDM4E
SCHEMBL7030548 0.74 SIRT6 (0.48) PARP1TYMPHSD17B10MAPTKDM4E
SCHEMBL7039377 0.74 PARP1 (0.53) PARP1TNKSHRH3CDK4CCND1
SCHEMBL21524690 0.74 PARP1 (0.53) PARP1TNKSHSD17B10HRH3CDK4
SCHEMBL349204 0.73 CHEK1 (0.53) PARP1TNKSCHEK1HSD17B10HRH3
SCHEMBL27683290 0.73 PARP1 (0.52) PARP1TNKSCHEK1HSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0878468-B1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL CO (JP) 2003-03-19 EP disclosed
EP-0775697-B1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL CO (JP) 2003-02-12 EP disclosed
US-5994542-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-11-30 US disclosed
EP-0878468-A1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-11-18 EP disclosed
US-5756738-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-05-26 US disclosed
EP-0775697-A1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-05-28 EP disclosed