SCHEMBL7024469

SCHEMBL7024469

COc1cccc(Cn2c(=O)c(C)c3sc(C(=O)O)cn3c2=O)c1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 15/20 0.58
FEN1 P39748 1/20 0.47
TP53 P04637 1/20 0.47
MAPT P10636 1/20 0.47
THRB P10828 1/20 0.47
ALDH1A1 P00352 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CMA1 P23946 1/20 0.45
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5957456 0.88 TRPA1 (0.72) TRPA1TP53MAPTALDH1A1
SCHEMBL5957675 0.86 TRPA1 (0.79) TRPA1TP53MAPT
SCHEMBL5957285 0.86 TRPA1 (0.76) TRPA1TP53
SCHEMBL6236419 0.85 TRPA1 (0.63) TRPA1TP53MAPT
SCHEMBL6238345 0.85 TRPA1 (0.62) TRPA1FEN1MAPTLMNA
SCHEMBL6237698 0.85 TRPA1 (0.60) TRPA1FEN1ALDH1A1
SCHEMBL6236549 0.83 TRPA1 (0.57) TRPA1FEN1
SCHEMBL5957429 0.82 TRPA1 (0.73) TRPA1ALDH1A1
SCHEMBL6234041 0.80 TRPA1 (0.59) TRPA1FEN1MAPTLMNA
SCHEMBL6235761 0.80 TRPA1 (0.56) TRPA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362054-A1 BICYCLIC PYRIMIDINE MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2003-11-19 EP disclosed
WO-2002064599-A1 BICYCLIC PYRIMIDINE MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO disclosed