SCHEMBL7024964

SCHEMBL7024964

NCCNc1ncc(-c2ncc[nH]2)c(-c2ccccc2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 7/20 0.46
MTOR P42345 1/20 0.43
ADK P55263 1/20 0.43
NISCH Q9Y2I1 1/20 0.43
GSK3B P49841 2/20 0.43
CCNB2 O95067 1/20 0.43
CDK1 P06493 1/20 0.43
CCNB1 P14635 1/20 0.43
GSK3A P49840 1/20 0.43
CCNB3 Q8WWL7 1/20 0.43
SYK P43405 2/20 0.39
ZAP70 P43403 1/20 0.39
CXCR4 P61073 1/20 0.36
PRKCZ Q05513 1/20 0.36
PRKD2 Q9BZL6 1/20 0.36
ADORA2A P29274 3/20 0.36
CSNK1A1 P48729 1/20 0.36
TYRO3 Q06418 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
PTGS2 P35354 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5089415 0.85 KDM1A (0.42) ADORA1GSK3BCCNB2CDK1CCNB1
SCHEMBL7024960 0.79 ADORA1 (0.48) ADORA1SYKZAP70ADORA2AKDM4E
SCHEMBL4992921 0.78 GSK3B (0.73) ADORA1MTORADKNISCHGSK3B
SCHEMBL27592597 0.77 GSK3B (0.55) ADORA1GSK3BCCNB2CDK1CCNB1
SCHEMBL27592588 0.73 GSK3B (0.49) ADORA1GSK3BCCNB2CDK1CCNB1
SCHEMBL14096954 0.73 GSK3B (0.58) ADORA1GSK3BCCNB2CDK1CCNB1
SCHEMBL14097003 0.73 GSK3B (0.51) ADORA1GSK3BCCNB2CDK1CCNB1
SCHEMBL27538052 0.73 GSK3B (0.40) ADORA1GSK3BCCNB2CDK1CCNB1
SCHEMBL5099784 0.73 GSK3B (0.43) ADORA1GSK3BCCNB2CDK1CCNB1
SCHEMBL5095053 0.72 GSK3B (0.50) ADORA1GSK3BCCNB2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317433-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2003-06-11 EP disclosed
WO-2002020495-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2002-03-14 WO disclosed
EP-1087963-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 Chiron Corporation (US) 2001-04-04 EP disclosed
WO-1999065897-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 1999-12-23 WO disclosed