SCHEMBL7026599

SCHEMBL7026599

O=c1[nH]c(=O)c2cccc(OCCCl)c2[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
DRD3 P35462 1/20 0.41
CCR1 P32246 1/20 0.39
KDM4E B2RXH2 3/20 0.39
CA12 O43570 1/20 0.39
PARP1 P09874 1/20 0.39
CA9 Q16790 1/20 0.39
ADORA3 P0DMS8 1/20 0.38
POLB P06746 2/20 0.37
HCAR2 Q8TDS4 3/20 0.36
HCAR3 P49019 1/20 0.36
GPR84 Q9NQS5 1/20 0.35
ALDH1A1 P00352 2/20 0.34
HPGD P15428 1/20 0.34
ALOX12 P18054 1/20 0.34
MAPK10 P53779 1/20 0.34
HSD17B10 Q99714 1/20 0.34
NQO2 P16083 1/20 0.34
ADRB2 P07550 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7025117 0.94 DRD2 (0.41) DRD2DRD4DRD3CCR1KDM4E
SCHEMBL7031280 0.88 PARP1 (0.41) DRD2DRD4DRD3CCR1KDM4E
SCHEMBL7040483 0.85 CYP2A6 (0.44) DRD2DRD4DRD3KDM4ECA12
SCHEMBL7030573 0.81 DAO (0.49) KDM4ECA12PARP1CA9ADORA3
SCHEMBL7032421 0.81 KDM4E (0.41) DRD2DRD4DRD3CCR1KDM4E
SCHEMBL7032366 0.78 CCR1 (0.43) DRD2DRD4DRD3CCR1KDM4E
SCHEMBL7031170 0.76 DRD2 (0.41) DRD2DRD4DRD3KDM4ECA12
SCHEMBL3423322 0.76 NQO2 (0.57) KDM4EPARP1POLBALDH1A1HPGD
SCHEMBL7030040 0.75 KDM4E (0.41) CCR1KDM4ECA12PARP1CA9
SCHEMBL7029217 0.75 KDM4E (0.41) KDM4ECA12PARP1CA9POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0878468-B1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL CO (JP) 2003-03-19 EP disclosed
EP-0775697-B1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL CO (JP) 2003-02-12 EP disclosed
US-5994542-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-11-30 US disclosed
EP-0878468-A1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-11-18 EP disclosed
US-5756738-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-05-26 US disclosed
EP-0775697-A1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-05-28 EP disclosed