SCHEMBL7027348

SCHEMBL7027348

COc1cccc(/C=C/C(=O)c2c(OC)cc(CO)c(C3=CCN(C)CC3)c2O)c1OC

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
ALOX5 P09917 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
NFE2L2 Q16236 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAOB P27338 2/20 0.42
ABCB1 P08183 1/20 0.41
CYP1A1 P04798 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
RELA Q04206 3/20 0.41
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
NTSR1 P30989 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7027485 0.92 ABCB1 (0.50) NPC1RAB9AALOX5SMN1; SMN2ABCB1
SCHEMBL746358 0.91 NPC1 (0.46) NPC1RAB9AALOX5L3MBTL1NFE2L2
SCHEMBL20858960 0.90 RAB9A (0.45) NPC1RAB9AALOX5L3MBTL1NFE2L2
SCHEMBL7027331 0.88 ABCG2 (0.49) NFE2L2MAOBALDH1A1
SCHEMBL7026486 0.86 MAPT (0.53) MAOBABCB1
SCHEMBL7028325 0.86 ABCB1 (0.48) L3MBTL1SMN1; SMN2ABCB1ALDH1A1LMNA
SCHEMBL7029021 0.85 ABCB1 (0.46) ABCB1
SCHEMBL7025959 0.85 AR (0.46) RAB9ASMN1; SMN2MAOBABCB1ALDH1A1
SCHEMBL7028079 0.85 ABCG2 (0.51) MAOBABCB1CYP1A2CYP2D6
SCHEMBL7027366 0.84 PDPK1 (0.47) ALOX5MAOBABCB1RELALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120121692-A1 COMPOUNDS AND COMPOSITIONS COMPRISING CDK INHIBITORS AND METHODS FOR TREATING CANCER SHANDONG UNIVERSITY (CN) 2012-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120121692-A1 COMPOUNDS AND COMPOSITIONS COMPRISING CDK INHIBITORS AND METHODS FOR TREATING CANCER CDK6, CDK5, CDK4 NPC1 3330/4885RAB9A 2710/4885ALOX5 2088/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.