SCHEMBL7028562

SCHEMBL7028562

O=c1[nH]c(=O)c2cc(CCCl)ccc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.47
CA9 Q16790 2/20 0.47
PARP1 P09874 4/20 0.46
KDM4E B2RXH2 3/20 0.46
SIRT6 Q8N6T7 2/20 0.41
SIRT2 Q8IXJ6 1/20 0.41
GAA P10253 1/20 0.41
PKM P14618 1/20 0.41
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PARG Q86W56 1/20 0.39
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PDE3A Q14432 2/20 0.37
GRIN2D O15399 2/20 0.36
GRIN3B O60391 2/20 0.36
GRIN1 Q05586 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7027027 0.87 PARP1 (0.46) CA12CA9PARP1KDM4EGAA
SCHEMBL7034143 0.86 CA12 (0.50) CA12CA9PARP1KDM4ESIRT6
SCHEMBL7033620 0.83 CA12 (0.47) CA12CA9PARP1KDM4ESIRT6
SCHEMBL6910223 0.82 GAA (0.59) GAAPKMALDH1A1MEN1MAPT
SCHEMBL7029630 0.82 KDM4E (0.53) CA12CA9PARP1KDM4ESIRT6
SCHEMBL7028337 0.79 CA12 (0.50) CA12CA9PARP1KDM4ESIRT6
SCHEMBL20942693 0.79 GAA (0.66) CA12CA9PARP1KDM4ESIRT6
SCHEMBL2056368 0.79 ALDH1A1 (0.50) CA12CA9PARP1KDM4EGAA
SCHEMBL7032932 0.79 CA12 (0.46) CA12CA9PARP1KDM4ESIRT6
SCHEMBL6273166 0.78 MAPT (0.46) PARP1KDM4EGAAALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0878468-B1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL CO (JP) 2003-03-19 EP disclosed
EP-0775697-B1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL CO (JP) 2003-02-12 EP disclosed
US-5994542-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-11-30 US disclosed
EP-0878468-A1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-11-18 EP disclosed
US-5756738-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-05-26 US disclosed
EP-0775697-A1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-05-28 EP disclosed