SCHEMBL7028635

SCHEMBL7028635

O=c1[nH]c(=O)c2cc(C(Cl)Cl)ccc2[nH]1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.50
CA9 Q16790 2/20 0.50
KDM4E B2RXH2 4/20 0.48
PARP1 P09874 2/20 0.48
ALDH1A1 P00352 2/20 0.42
HPGD P15428 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PARG Q86W56 1/20 0.40
PDE3A Q14432 5/20 0.39
NAPEPLD Q6IQ20 1/20 0.37
PDE3B Q13370 3/20 0.37
TYMP P19971 2/20 0.35
GSK3B P49841 1/20 0.35
BACE1 P56817 1/20 0.35
SIRT6 Q8N6T7 2/20 0.34
GAA P10253 1/20 0.34
GRIA1 P42261 1/20 0.33
CACNG8 Q8WXS5 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7032963 0.86 CA12 (0.47) CA12CA9KDM4EPARP1ALDH1A1
SCHEMBL7035473 0.86 PARP1 (0.48) CA12CA9KDM4EPARP1ALDH1A1
SCHEMBL7026218 0.83 CA12 (0.45) CA12CA9KDM4EPARP1ALDH1A1
SCHEMBL9761076 0.82 KDM4E (0.50) CA12CA9KDM4EPARP1ALDH1A1
SCHEMBL7030965 0.82 KDM4E (0.50) CA12CA9KDM4EPARP1ALDH1A1
SCHEMBL404118 0.76 PARP1 (0.56) CA12CA9KDM4EPARP1ALDH1A1
SCHEMBL7032932 0.75 CA12 (0.46) CA12CA9KDM4EPARP1ALDH1A1
SCHEMBL7029487 0.75 CA12 (0.46) CA12CA9KDM4EPARP1ALDH1A1
SCHEMBL3772977 0.74 PARP1 (0.55) CA12CA9KDM4EPARP1ALDH1A1
Potassium SCHEMBL3643814 0.74 PARP1 (0.55) CA12CA9KDM4EPARP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0878468-B1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL CO (JP) 2003-03-19 EP disclosed
EP-0775697-B1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL CO (JP) 2003-02-12 EP disclosed
US-5994542-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-11-30 US disclosed
EP-0878468-A1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-11-18 EP disclosed
US-5756738-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-05-26 US disclosed
EP-0775697-A1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-05-28 EP disclosed