SCHEMBL7029072

SCHEMBL7029072

Cc1c[nH]c(-c2ccc(N)nc2-c2ccc(Cl)cc2Cl)n1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.45
HSP90AB1 P08238 2/20 0.45
DPP4 P27487 5/20 0.39
CNR1 P21554 3/20 0.37
CNR2 P34972 3/20 0.37
HSD11B1 P28845 1/20 0.37
CRHR1 P34998 5/20 0.36
LMNA P02545 1/20 0.36
CYP3A4 P08684 1/20 0.35
MAP3K14 Q99558 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27538173 0.84 MAP3K14 (0.48) HSP90AA1HSP90AB1DPP4LMNAMAP3K14
SCHEMBL7852616 0.78 GSK3B (0.47) HSP90AA1HSP90AB1DPP4CNR1CNR2
SCHEMBL29438549 0.77 NPSR1 (0.39) HSP90AA1HSP90AB1HSD11B1CRHR1MAP3K14
SCHEMBL4975912 0.76 HSP90AA1 (0.36) HSP90AA1HSP90AB1HSD11B1CRHR1
SCHEMBL3660492 0.76 CYP3A4 (0.43) HSP90AA1HSP90AB1LMNACYP3A4
SCHEMBL3317224 0.75 ALDH1A1 (0.50) HSP90AA1HSP90AB1HSD11B1CRHR1
SCHEMBL952939 0.74 HSP90AA1 (0.37) HSP90AA1HSP90AB1CNR1CNR2HSD11B1
SCHEMBL31429725 0.74 IDO1 (0.41) HSP90AA1HSP90AB1CYP3A4
SCHEMBL13257647 0.73 HSP90AA1 (0.36) HSP90AA1HSP90AB1DPP4CNR1CNR2
SCHEMBL4399097 0.73 GSK3B (0.64) HSP90AA1HSP90AB1DPP4HSD11B1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317433-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2003-06-11 EP disclosed
WO-2002020495-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2002-03-14 WO disclosed