SCHEMBL7029520

SCHEMBL7029520

O=c1[nH]c(=O)c2cccc(CBr)c2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.44
KDM4E B2RXH2 3/20 0.44
CA12 O43570 1/20 0.44
CA9 Q16790 1/20 0.44
ALDH1A1 P00352 3/20 0.41
TYMP P19971 2/20 0.35
GSK3B P49841 1/20 0.35
BACE1 P56817 1/20 0.35
DAO P14920 2/20 0.34
LMNA P02545 4/20 0.34
FEN1 P39748 1/20 0.34
MEN1 O00255 2/20 0.33
POLB P06746 2/20 0.33
BLM P54132 2/20 0.33
KMT2A Q03164 2/20 0.33
GDA Q9Y2T3 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
DHODH Q02127 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2914712 0.84 ALDH1A1 (0.49) PARP1KDM4ECA12CA9ALDH1A1
SCHEMBL7032649 0.82 PARP1 (0.44) PARP1KDM4ECA12CA9ALDH1A1
SCHEMBL7030918 0.79 DAO (0.48) PARP1KDM4ECA12CA9ALDH1A1
SCHEMBL7027616 0.79 PARP1 (0.42) PARP1KDM4ECA12CA9ALDH1A1
SCHEMBL24262307 0.78 FEN1 (0.57) PARP1KDM4ECA12CA9ALDH1A1
SCHEMBL7033769 0.78 GAA (0.42) PARP1KDM4ECA12CA9ALDH1A1
SCHEMBL7030625 0.78 PARP1 (0.41) PARP1KDM4ECA12CA9ALDH1A1
SCHEMBL2731038 0.76 PARP1 (0.48) PARP1KDM4ECA12CA9TYMP
SCHEMBL7032421 0.75 KDM4E (0.41) PARP1KDM4ECA12CA9ALDH1A1
SCHEMBL2919116 0.72 CHEK1 (0.53) PARP1KDM4ECA12CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0878468-B1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL CO (JP) 2003-03-19 EP disclosed
EP-0775697-B1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL CO (JP) 2003-02-12 EP disclosed
US-5994542-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-11-30 US disclosed
EP-0878468-A1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-11-18 EP disclosed
US-5756738-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-05-26 US disclosed
EP-0775697-A1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-05-28 EP disclosed