SCHEMBL7030282

SCHEMBL7030282

CN1CCN(c2cccc3c2C[C@H](NC(=O)c2cccc(C(F)(F)F)c2)CC3)CC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
KCNH2 Q12809 4/20 0.49
SCN9A Q15858 4/20 0.49
SCN5A Q14524 3/20 0.49
MTNR1A P48039 1/20 0.48
MTNR1B P49286 1/20 0.48
TAS1R3 Q7RTX0 1/20 0.47
TAS1R1 Q7RTX1 1/20 0.47
TAS1R2 Q8TE23 1/20 0.47
BRAF P15056 1/20 0.46
DRD2 P14416 1/20 0.46
DRD1 P21728 1/20 0.46
HDAC8 Q9BY41 2/20 0.45
PAK1 Q13153 1/20 0.45
PHGDH O43175 1/20 0.44
JAK2 O60674 1/20 0.44
SRC P12931 1/20 0.44
CHRM4 P08173 1/20 0.44
CHRM5 P08912 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7031232 1.00 MEN1 (0.55) MEN1KMT2AKCNH2SCN9ASCN5A
SCHEMBL4788895 0.93 KCNH2 (0.49) MEN1KMT2AKCNH2SCN9ASCN5A
SCHEMBL6820338 0.91 KCNH2 (0.55) MEN1KMT2AKCNH2SCN9ASCN5A
SCHEMBL7025761 0.91 KCNH2 (0.55) MEN1KMT2AKCNH2SCN9ASCN5A
SCHEMBL6820334 0.91 KCNH2 (0.55) MEN1KMT2AKCNH2SCN9ASCN5A
SCHEMBL7026344 0.86 MTNR1A (0.52) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL7026340 0.86 MTNR1A (0.52) KCNH2SCN9ASCN5AMTNR1AMTNR1B
SCHEMBL4789479 0.86 LCK (0.46) MEN1KMT2AKCNH2SCN9ASCN5A
SCHEMBL4789251 0.86 KCNH2 (0.45) MEN1KMT2AKCNH2SCN9ASCN5A
SCHEMBL4789031 0.86 KCNH2 (0.47) MEN1KMT2AKCNH2SCN9ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002022738-A9 SPECIES MODIFICATION IN MACROCYCLIC POLYESTER OLIGOMERS, AND COMPOSITIONS PREPARED THEREBY CYCLICS CORP (US) 2003-03-27 WO disclosed
EP-0888319-B1 SUBSTITUTED 1,2,3,4-TETRAHYDRONAPHTHALENE DERIVATIVES ASTRAZENECA AB (SE) 2003-01-29 EP disclosed
US-6410530-B1 CENTRAL NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS ASTRAZENECA AB (SE) 2002-06-25 US disclosed
US-6124283-A Substituted 1,2,3,4-tetrahydronaphthalene derivatives ASTRA AKTIEBOLAG (SE) 2000-09-26 US disclosed