SCHEMBL7035641

SCHEMBL7035641

CC(C)(C)Sc1ccccc1-c1ccccn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.45
LMNA P02545 4/20 0.45
CCR1 P32246 2/20 0.45
CCR5 P51681 2/20 0.45
CCR8 P51685 2/20 0.45
CYP1A2 P05177 1/20 0.45
POLB P06746 1/20 0.45
METAP1 P53582 1/20 0.45
BLM P54132 1/20 0.45
HIF1A Q16665 1/20 0.45
DOHH Q9BU89 1/20 0.45
P4HTM Q9NXG6 1/20 0.45
NPC1 O15118 7/20 0.44
RAB9A P51151 6/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
L3MBTL1 Q9Y468 4/20 0.44
TP53 P04637 3/20 0.44
HTT P42858 3/20 0.44
ALOX15 P16050 2/20 0.44
PKM P14618 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30093761 0.85 GRM5 (0.39) KDM4ELMNACCR1CCR5CCR8
SCHEMBL5919364 0.82 KDM4E (0.45) KDM4ELMNACCR1CCR5CCR8
SCHEMBL1207426 0.79 KDM4E (0.50) KDM4ELMNACCR1CCR5CCR8
SCHEMBL31038172 0.79 KDM4E (0.50) KDM4ELMNACCR1CCR5CCR8
SCHEMBL28087696 0.79 KDM4E (0.54) KDM4ELMNACCR1CCR5CCR8
SCHEMBL11605127 0.76 KDM4E (0.50) KDM4ELMNACCR1CCR5CCR8
SCHEMBL11140262 0.74 KDM4E (0.48) KDM4ELMNACCR1CCR5CCR8
SCHEMBL28087698 0.74 KDM4E (0.48) KDM4ELMNACCR1CCR5CCR8
SCHEMBL858806 0.73 KDM4E (0.72) KDM4ELMNACCR1CCR5CCR8
SCHEMBL5322670 0.73 KDM4E (0.46) KDM4ELMNACCR1CCR5CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003055477-A1 METHOD FOR THE TREATMENT OF MC RECEPTOR RELATED DISORDERS WITH A CHELATE AND/OR A CHELATOR 7TM PHARMA A/S (DK) 2003-07-10 WO disclosed
WO-2003003008-A1 CHEMICAL LIBRARIES USEFUL FOR DRUG DISCOVERY PROCESSES 7TM PHARMA A/S (DK) 2003-01-09 WO disclosed
WO-2003003009-A1 USE OF METAL-ION CHELATES IN VALIDATING BIOLOGICAL MOLECULES AS DRUG TARGETS IN TEST ANIMAL MODELS 7TM PHARMA A/S (DK) 2003-01-09 WO disclosed