SCHEMBL7040495

SCHEMBL7040495

CCCN1CCC(c2nc3c(OC(N)=O)cccc3n2C)C1

nearest known ligand 0.65

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.65
PARP2 Q9UGN5 1/20 0.44
DRD2 P14416 2/20 0.41
DRD3 P35462 2/20 0.41
KDM2B Q8NHM5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7044350 0.91 PARP1 (0.53) PARP1PARP2DRD2DRD3KDM2B
SCHEMBL7042319 0.89 PARP1 (0.52) PARP1PARP2DRD2DRD3KDM2B
SCHEMBL7035297 0.89 PARP1 (0.52) PARP1PARP2DRD2DRD3KDM2B
SCHEMBL7038527 0.89 PARP1 (0.52) PARP1DRD3
SCHEMBL7042136 0.88 PARP1 (0.51) PARP1PARP2DRD2DRD3KDM2B
SCHEMBL7045627 0.88 PARP1 (0.50) PARP1PARP2DRD2DRD3KDM2B
SCHEMBL7043782 0.88 PARP1 (0.52) PARP1PARP2DRD2DRD3KDM2B
SCHEMBL7040671 0.87 PARP1 (0.50) PARP1PARP2
SCHEMBL7041082 0.87 PARP1 (0.52) PARP1DRD2
SCHEMBL7039404 0.87 PARP1 (0.49) PARP1PARP2DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed