SCHEMBL7040671

SCHEMBL7040671

CN1CCC(c2nc3c(OC(N)=O)cccc3n2C)C1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.50
HSD11B1 P28845 1/20 0.41
PARP2 Q9UGN5 3/20 0.40
HTR2B P41595 1/20 0.39
KCNH2 Q12809 6/20 0.36
CHRM1 P11229 3/20 0.36
HRH1 P35367 3/20 0.36
CYP2D6 P10635 2/20 0.36
HTR6 P50406 1/20 0.36
PROKR1 Q8TCW9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7040201 0.93 PARP1 (0.54) PARP1HSD11B1PARP2HTR2BCHRM1
SCHEMBL7038340 0.88 PARP1 (0.48) PARP1HSD11B1HTR2BPROKR1
SCHEMBL7040495 0.87 PARP1 (0.65) PARP1PARP2
SCHEMBL7043780 0.87 PARP1 (0.47) PARP1HSD11B1PARP2HTR2BKCNH2
SCHEMBL7044945 0.85 PARP1 (0.45) PARP1HSD11B1HTR2BPROKR1
SCHEMBL7045615 0.85 PARP1 (0.51) PARP1PARP2HTR2BKCNH2CYP2D6
SCHEMBL7041082 0.85 PARP1 (0.52) PARP1HTR2BHTR6
SCHEMBL7042003 0.83 PARP1 (0.48) PARP1PARP2HTR2B
SCHEMBL5621671 0.83 PARP1 (0.71) PARP1PARP2
SCHEMBL7038527 0.82 PARP1 (0.52) PARP1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed