SCHEMBL7042936

SCHEMBL7042936

CCCN1CCCN(c2nc3c(OC(N)=O)cccc3n2C(C)C)CC1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PARP1 P09874 2/20 0.38
ALDH1A1 P00352 3/20 0.37
HTT P42858 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
DRD2 P14416 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7038476 0.96 MEN1 (0.40) MEN1KMT2APARP1ALDH1A1HTT
SCHEMBL7038533 0.89 PARP1 (0.47) PARP1ALDH1A1DRD2L3MBTL1
SCHEMBL7043633 0.87 PARP1 (0.41) MEN1KMT2APARP1ALDH1A1CYP1A2
SCHEMBL7043857 0.86 ALDH1A1 (0.43) MEN1KMT2APARP1ALDH1A1
SCHEMBL5619750 0.86 PARP1 (0.52) MEN1KMT2APARP1ALDH1A1HTT
SCHEMBL7039979 0.85 PARP1 (0.50) MEN1KMT2APARP1DRD2L3MBTL1
SCHEMBL7040070 0.85 NPSR1 (0.40) MEN1KMT2APARP1ALDH1A1
SCHEMBL7047366 0.85 NPSR1 (0.40) MEN1KMT2APARP1ALDH1A1
SCHEMBL7041749 0.85 ALDH1A1 (0.44) MEN1KMT2APARP1ALDH1A1SMN1; SMN2
SCHEMBL7043577 0.84 ALDH1A1 (0.44) MEN1KMT2APARP1ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed