SCHEMBL7044630

SCHEMBL7044630

CCCN1CCCC1c1nc2c(OC(N)=O)cccc2n1CCN(C)C

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.41
HTR2A P28223 4/20 0.36
DRD1 P21728 4/20 0.36
SCN9A Q15858 1/20 0.35
DRD2 P14416 4/20 0.35
HTR1A P08908 3/20 0.34
BRD4 O60885 2/20 0.33
CREBBP Q92793 2/20 0.33
CYP2D6 P10635 1/20 0.33
HRH1 P35367 1/20 0.33
KCNH2 Q12809 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33
OPRL1 P41146 1/20 0.33
OGFRL1 Q5TC84 1/20 0.33
HIF1A Q16665 1/20 0.33
TP53 P04637 1/20 0.33
ADORA2A P29274 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7042328 0.90 PARP1 (0.43) PARP1HTR2ADRD1SCN9ADRD2
SCHEMBL7041865 0.90 PARP1 (0.43) PARP1HTR2ADRD1SCN9ADRD2
SCHEMBL7045984 0.90 PARP1 (0.44) PARP1HTR2ADRD1SCN9ADRD2
SCHEMBL7044198 0.89 PARP1 (0.42) PARP1HTR2ADRD1SCN9ADRD2
SCHEMBL7045077 0.88 PARP1 (0.44) PARP1HTR2ADRD1SCN9ADRD2
SCHEMBL5622204 0.86 PARP1 (0.55) PARP1HTR1A
SCHEMBL7041326 0.85 PARP1 (0.43) PARP1HTR2ASCN9ADRD2CYP2D6
SCHEMBL7043521 0.85 PARP1 (0.45) PARP1DRD2CYP2D6HRH1KCNH2
SCHEMBL7041972 0.85 PARP1 (0.55) PARP1DRD2BRD4CREBBPHRH1
SCHEMBL7039404 0.84 PARP1 (0.49) PARP1DRD2BRD4CREBBPCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed