SCHEMBL7044663

SCHEMBL7044663

NC(=O)Oc1cccc2c1nc(C1CCCNC1)n2CCN1CCCCC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 3/20 0.44
HRH1 P35367 2/20 0.44
NPY1R P25929 7/20 0.42
PARP1 P09874 6/20 0.38
MEN1 O00255 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38
PKM P14618 1/20 0.38
HPGD P15428 1/20 0.38
PARP2 Q9UGN5 4/20 0.37
PARP3 Q9Y6F1 3/20 0.37
TNKS O95271 1/20 0.37
CHRM2 P08172 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
ADRA1A P35348 1/20 0.37
SLC6A3 Q01959 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7042453 0.99 CHRM1 (0.44) CHRM1HRH1NPY1RPARP1MEN1
SCHEMBL7042033 0.95 NPY1R (0.40) CHRM1HRH1NPY1RPARP1MEN1
SCHEMBL7042457 0.95 JAK2 (0.39) CHRM1HRH1NPY1RPARP1MEN1
SCHEMBL7040421 0.90 JAK2 (0.44) HRH1NPY1RPARP1MEN1CYP3A4
SCHEMBL7043993 0.89 CHRM1 (0.46) CHRM1HRH1NPY1RPARP1PARP2
SCHEMBL7041213 0.89 CHRM1 (0.46) CHRM1HRH1NPY1RPARP1PARP2
SCHEMBL7045696 0.86 CHRM1 (0.48) CHRM1HRH1NPY1RPARP1PARP2
SCHEMBL5621194 0.86 PARP1 (0.53) CHRM1HRH1PARP1MEN1CYP3A4
SCHEMBL7040702 0.86 KMT2A (0.42) NPY1RPARP1MEN1CYP3A4CYP2D6
SCHEMBL7044486 0.86 CHRM1 (0.44) CHRM1HRH1NPY1RPARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed