Choline

Choline

SCHEMBL7044734

C[N+](C)(C)CCO.Oc1c[nH]c2ccccc12

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3GNRHRMPLPDE3APDE3BPDE4APDE4BPDE4CPDE4DPPARASLC5A2

The experimentally established mechanism targets of Choline. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
GPR84 Q9NQS5 2/20 0.44
MAPT P10636 1/20 0.44
AHR P35869 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
PBRM1 Q86U86 1/20 0.44
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 3/20 0.43
MAPK1 P28482 1/20 0.43
POLB P06746 1/20 0.43
GAA P10253 1/20 0.43
CYP2D6 P10635 2/20 0.42
CYP2C19 P33261 2/20 0.42
HSD17B10 Q99714 2/20 0.42
TSHR P16473 1/20 0.42
ATM Q13315 1/20 0.42
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Choline SCHEMBL1938782 0.90 POLB (0.42) CYP3A4MEN1KMT2AGPR84MAPT
SCHEMBL27815030 0.81 MAPT (0.39) CYP3A4MEN1KMT2AGPR84MAPT
SCHEMBL155191 0.80 MEN1 (0.58) CYP3A4MEN1KMT2AGPR84MAPT
SCHEMBL29567690 0.80 MEN1 (0.58) CYP3A4MEN1KMT2AGPR84MAPT
SCHEMBL28624457 0.78 MEN1 (0.56) CYP3A4MEN1KMT2AGPR84MAPT
Methane SCHEMBL5065725 0.78 MEN1 (0.56) CYP3A4MEN1KMT2AGPR84MAPT
SCHEMBL10550137 0.78 MEN1 (0.56) CYP3A4MEN1KMT2AGPR84MAPT
Hydrochloric Acid SCHEMBL28628671 0.78 MEN1 (0.56) CYP3A4MEN1KMT2AGPR84MAPT
Water SCHEMBL27616945 0.78 MEN1 (0.56) CYP3A4MEN1KMT2AGPR84MAPT
SCHEMBL27702719 0.78 MEN1 (0.56) CYP3A4MEN1KMT2AGPR84MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1219628-B1 Novel substrates for detection of microbial metabolites BIOSYNTH AG (CH) 2003-04-02 EP claimed