SCHEMBL7045124

SCHEMBL7045124

NC(=O)Oc1cc(N)cc2[nH]c(C3CCNC3)nc12

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 18/20 0.53
PARP2 Q9UGN5 2/20 0.40
PBK Q96KB5 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
GFER P55789 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7042529 0.93 PARP1 (0.54) PARP1PARP2PBKKDM4EMAPT
SCHEMBL7038859 0.93 PARP1 (0.51) PARP1PARP2PBKKDM4EMAPT
SCHEMBL7040921 0.88 PARP1 (0.52) PARP1PARP2
SCHEMBL7043271 0.85 PARP1 (0.49) PARP1PARP2
SCHEMBL7042400 0.83 PARP1 (0.47) PARP1PARP2
SCHEMBL6869625 0.83 PARP1 (0.69) PARP1PARP2
SCHEMBL5621403 0.82 PARP1 (0.69) PARP1PARP2
SCHEMBL7040577 0.81 PARP1 (0.54) PARP1PARP2PBK
SCHEMBL7042256 0.81 PARP1 (0.51) PARP1PARP2PBK
SCHEMBL7040728 0.79 PARP1 (0.51) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed