SCHEMBL7045165

SCHEMBL7045165

COc1cccc(C(O)(C(C)C)C(C)CN(C)C)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP2C19 P33261 1/20 0.48
HSD17B10 Q99714 1/20 0.48
AOC3 Q16853 2/20 0.42
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
CYP3A4 P08684 1/20 0.38
HIF1A Q16665 1/20 0.38
HTR2A P28223 3/20 0.38
KCNH2 Q12809 2/20 0.38
OPRM1 P35372 2/20 0.38
OPRD1 P41143 2/20 0.38
MRGPRX2 Q96LB1 1/20 0.38
CHRM3 P20309 1/20 0.38
HRH2 P25021 1/20 0.38
ADRA1A P35348 1/20 0.38
OPRK1 P41145 1/20 0.38
TAAR1 Q96RJ0 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8687121 0.99 CYP2D6 (0.47) CYP2D6ALDH1A1CYP2C19HSD17B10AOC3
SCHEMBL7591195 0.86 CYP2D6 (0.62) CYP2D6ALDH1A1CYP2C19HSD17B10AOC3
SCHEMBL7591201 0.86 CYP2D6 (0.62) CYP2D6ALDH1A1CYP2C19HSD17B10AOC3
SCHEMBL10350134 0.85 CYP17A1 (0.46) CYP2D6ALDH1A1CYP2C19HSD17B10AOC3
Hydrochloric Acid SCHEMBL8014032 0.84 CYP2D6 (0.60) CYP2D6ALDH1A1CYP2C19HSD17B10AOC3
SCHEMBL8529142 0.84 CYP2D6 (0.49) CYP2D6ALDH1A1CYP2C19HSD17B10AOC3
SCHEMBL169116 0.84 CYP2D6 (0.49) CYP2D6ALDH1A1CYP2C19HSD17B10AOC3
SCHEMBL355959 0.84 CYP2D6 (0.49) CYP2D6ALDH1A1CYP2C19HSD17B10AOC3
Hydrochloric Acid SCHEMBL8014025 0.84 CYP2D6 (0.60) CYP2D6ALDH1A1CYP2C19HSD17B10AOC3
Hydrochloric Acid SCHEMBL8686514 0.83 CYP2D6 (0.48) CYP2D6ALDH1A1CYP2C19HSD17B10AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0983995-B1 Pharmaceutically-active dimethyl-(3-aryl-but-3-enyl)-amine compounds GRUENENTHAL GMBH (DE) 2004-03-31 EP disclosed
EP-1069106-B1 Dimethyl-(3-aryl-but-3-enyl) amine derivatives with analgesic activity GRUENENTHAL GMBH (DE) 2004-01-28 EP disclosed
EP-0799819-B1 1-Dimethylaminomethyl 2-phenyl cycloalk-2-ene derivatives with analgesic activity GRUENENTHAL GMBH (DE) 2002-09-11 EP disclosed
EP-1069106-A2 Dimethyl-(3-aryl-but-3-enyl) amine derivatives with analgesic activity Grünenthal GmbH (DE) 2001-01-17 EP disclosed
EP-0983995-A2 Pharmaceutically-active dimethyl-(3-aryl-but-3-enyl)-amine compounds Grünenthal GmbH (DE) 2000-03-08 EP disclosed
EP-0799819-A1 Dimethyl-(3-aryl-but-3-enyl) amine derivatives with analgesic activity Grünenthal GmbH (DE) 1997-10-08 EP disclosed