SCHEMBL10350134

SCHEMBL10350134

COc1ccc2cc(C(O)(C(C)C)C(C)CN(C)C)ccc2c1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.46
ABCB11 O95342 1/20 0.41
ALDH1A1 P00352 2/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GAA P10253 1/20 0.39
CYP3A4 P08684 1/20 0.38
PTGS2 P35354 3/20 0.38
PTGS1 P23219 2/20 0.38
AKR1C3 P42330 2/20 0.38
AKR1C2 P52895 2/20 0.38
CDC42 P60953 1/20 0.38
RAC1 P63000 1/20 0.38
CYP1A2 P05177 1/20 0.38
TSHR P16473 1/20 0.38
SLC22A6 Q4U2R8 1/20 0.38
AOC3 Q16853 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10349478 0.88 ALDH1A1 (0.39) CYP17A1ALDH1A1CYP2D6CYP2C19HSD17B10
SCHEMBL7045165 0.85 CYP2D6 (0.48) ALDH1A1CYP2D6CYP2C19HSD17B10CYP3A4
SCHEMBL10349820 0.85 HIF1A (0.38) CYP17A1ALDH1A1CYP2D6CYP2C19HSD17B10
Hydrochloric Acid SCHEMBL8687121 0.84 CYP2D6 (0.47) ALDH1A1CYP2D6CYP2C19HSD17B10CYP3A4
SCHEMBL10868854 0.81 ALDH1A1 (0.47) CYP17A1ABCB11ALDH1A1CYP2D6CYP2C19
SCHEMBL10349821 0.79 CYP17A1 (0.44) CYP17A1ABCB11ALDH1A1CYP3A4PTGS2
SCHEMBL17775051 0.73 CYP17A1 (0.55) CYP17A1ABCB11CYP3A4PTGS2PTGS1
SCHEMBL10869652 0.73 ALDH1A1 (0.40) CYP17A1ALDH1A1CYP2D6CYP2C19HSD17B10
SCHEMBL11874066 0.73 CYP17A1 (0.44) CYP17A1ABCB11ALDH1A1CYP3A4PTGS2
SCHEMBL7043342 0.71 ALDH1A1 (0.48) ALDH1A1CYP2D6CYP2C19HSD17B10GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0176049-B1 AMINOALKYLNAPHTALENE DERIVATIVES HAVING PHARMACOLOGICAL ACTIVITIES CONSIGLIO NAZIONALE DELLE RICERCHE (IT) 1990-06-13 EP disclosed
EP-0176049-A2 Aminoalkylnaphtalene derivatives having pharmacological activities CONSIGLIO NAZIONALE DELLE RICERCHE (IT) 1986-04-02 EP disclosed