SCHEMBL7046897

SCHEMBL7046897

CCCN1CCCC(c2nc3c(OC(N)=O)cccc3n2CC)C1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.48
DRD3 P35462 4/20 0.43
ACHE P22303 1/20 0.42
KDM2B Q8NHM5 1/20 0.42
SIGMAR1 Q99720 3/20 0.41
DRD4 P21917 3/20 0.41
DRD2 P14416 2/20 0.41
NFKB1 P19838 1/20 0.41
PRCP P42785 1/20 0.41
EBP Q15125 1/20 0.41
DRD1 P21728 1/20 0.41
DRD5 P21918 1/20 0.41
CYP2D6 P10635 2/20 0.40
HRH1 P35367 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7044350 0.95 PARP1 (0.53) PARP1DRD3KDM2BDRD2HRH1
SCHEMBL7042194 0.93 PARP1 (0.47) PARP1DRD3ACHEKDM2BSIGMAR1
SCHEMBL7045127 0.93 PARP1 (0.47) PARP1DRD3ACHEKDM2BSIGMAR1
SCHEMBL7043437 0.93 PARP1 (0.49) PARP1DRD3ACHEKDM2BSIGMAR1
SCHEMBL7043532 0.92 PARP1 (0.48) PARP1DRD3ACHEKDM2BSIGMAR1
SCHEMBL7043338 0.90 PARP1 (0.59) PARP1DRD2HRH1
SCHEMBL7043521 0.90 PARP1 (0.45) PARP1DRD3ACHEKDM2BSIGMAR1
SCHEMBL7043782 0.90 PARP1 (0.52) PARP1DRD3ACHEKDM2BDRD2
SCHEMBL7042142 0.89 PARP1 (0.52) PARP1DRD3ACHEKDM2BDRD2
SCHEMBL7035297 0.88 PARP1 (0.52) PARP1DRD3KDM2BDRD2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed