3-Formylindole

3-Formylindole

SCHEMBL7048099

O=C(O)C(F)(F)F.O=Cc1c[nH]c2ccccc12

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.72
IMPDH2 P12268 1/20 0.72
MAPK1 P28482 2/20 0.54
HPGD P15428 4/20 0.52
ALDH1A1 P00352 4/20 0.52
MEN1 O00255 4/20 0.52
MAPT P10636 4/20 0.52
KMT2A Q03164 4/20 0.52
NPC1 O15118 3/20 0.52
RAB9A P51151 3/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
NFKB1 P19838 1/20 0.52
NFKB2 Q00653 1/20 0.52
RELA Q04206 1/20 0.52
HTT P42858 1/20 0.49
PIM1 P11309 1/20 0.47
PIM3 Q86V86 1/20 0.47
PIM2 Q9P1W9 1/20 0.47
PTGS2 P35354 1/20 0.46
APP P05067 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
3-Formylindole SCHEMBL28119225 0.85 CYP2A6 (0.79) CYP2A6IMPDH2MAPK1HPGDALDH1A1
3-Formylindole SCHEMBL30782674 0.85 CYP2A6 (1.00) CYP2A6IMPDH2HPGDALDH1A1MEN1
3-Formylindole SCHEMBL38654556 0.85 CYP2A6 (1.00) CYP2A6IMPDH2HPGDALDH1A1MEN1
3-Formylindole SCHEMBL30786737 0.85 CYP2A6 (1.00) CYP2A6IMPDH2HPGDALDH1A1MEN1
3-Formylindole SCHEMBL56373 0.85 CYP2A6 (1.00) CYP2A6IMPDH2HPGDALDH1A1MEN1
3-Formylindole SCHEMBL23630272 0.83 CYP2A6 (0.96) CYP2A6IMPDH2HPGDALDH1A1MEN1
3-Formylindole SCHEMBL30234679 0.83 CYP2A6 (0.96) CYP2A6IMPDH2HPGDALDH1A1MEN1
3-Formylindole SCHEMBL7432698 0.83 CYP2A6 (0.96) CYP2A6IMPDH2HPGDALDH1A1MEN1
3-Formylindole SCHEMBL27637265 0.83 CYP2A6 (0.96) CYP2A6IMPDH2HPGDALDH1A1MEN1
3-Formylindole SCHEMBL27269605 0.83 CYP2A6 (0.96) CYP2A6IMPDH2HPGDALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1476151-A1 1-ARYLSULFONYL-3-SUBSTITUED INDOLE AND INDOLINE DERIVATES USEFUL IN THE TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS Akzo Nobel N.V. (NL) 2004-11-17 EP disclosed
WO-2003068220-A1 1-ARYLSULFONYL-3-SUBSTITUTED INDOLE AND INDOLINE DERIVATIVES USEFUL IN THE TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS AKZO NOBEL N.V. (NL) 2003-08-21 WO disclosed