SCHEMBL7050488

SCHEMBL7050488

NC(=O)c1ccc2nc(CCc3ccccc3)[nH]c2c1

nearest known ligand 0.73

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.73
RAB9A P51151 2/20 0.65
ALDH1A1 P00352 2/20 0.65
MAPT P10636 1/20 0.65
SMN1; SMN2 Q16637 1/20 0.65
CHEK2 O96017 7/20 0.60
NPC1 O15118 1/20 0.58
HDAC1 Q13547 1/20 0.57
APEX1 P27695 1/20 0.56
NPSR1 Q6W5P4 1/20 0.52
F2 P00734 1/20 0.51
F10 P00742 1/20 0.51
F7 P08709 1/20 0.51
MAPK1 P28482 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6374801 0.91 HDAC6 (0.62) HDAC6RAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL7050481 0.90 HDAC6 (0.59) HDAC6RAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL18229598 0.85 HDAC6 (1.00) HDAC6RAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL6374805 0.81 HDAC6 (0.51) HDAC6RAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL14347041 0.79 CHEK2 (0.60) CHEK2APEX1NPSR1F2F10
SCHEMBL6368278 0.78 KDM4E (0.52) HDAC6ALDH1A1CHEK2APEX1NPSR1
SCHEMBL4657967 0.77 HDAC6 (0.60) HDAC6RAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL20085778 0.77 GAA (0.68) HDAC6ALDH1A1MAPTSMN1; SMN2HDAC1
SCHEMBL6367630 0.77 HDAC6 (0.59) HDAC6RAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL8974004 0.76 KMT2A (0.77) HDAC6RAB9AALDH1A1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003024451-A1 2-(2-PHENYLETHYL)-BENZIMIDAZOLE-5-CARBOXAMIDE DERIVATIVES AND THEIR USE AS TRYPTASE INHIBITORS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2003-03-27 WO disclosed