SCHEMBL7051101

SCHEMBL7051101

CC(=O)ON=C1C(=O)Nc2cc(Cl)c([N+](=O)[O-])c(Cl)c2C1=O

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
TSHR P16473 2/20 0.33
POLB P06746 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
MPI P34949 1/20 0.31
BLM P54132 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CES1 P23141 2/20 0.31
CCNB2 O95067 2/20 0.30
CDK1 P06493 2/20 0.30
CCNB1 P14635 2/20 0.30
GSK3A P49840 2/20 0.30
GSK3B P49841 2/20 0.30
CDK5 Q00535 2/20 0.30
CDK5R1 Q15078 2/20 0.30
CCNB3 Q8WWL7 2/20 0.30
UCHL3 P15374 1/20 0.30
UCHL1 P09936 1/20 0.30
DCTPP1 Q9H773 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7054500 0.91 TSHR (0.36) ALDH1A1TSHRPOLBGAAMAPT
SCHEMBL7050080 0.91 CES1 (0.33) ALDH1A1TSHRCES1CCNB2CDK1
SCHEMBL7048302 0.85 CES1 (0.36) CES1CCNB2CDK1CCNB1GSK3A
SCHEMBL7052308 0.84 TSHR (0.36) ALDH1A1TSHRCES1CCNB2CDK1
SCHEMBL7049385 0.84 MAPT (0.38) ALDH1A1POLBGAAMAPTMPI
SCHEMBL7051585 0.83 TSHR (0.34) ALDH1A1TSHRCES1CCNB2CDK1
SCHEMBL7048408 0.82 TSHR (0.39) ALDH1A1TSHRPOLBGAAMAPT
SCHEMBL7048406 0.82 TSHR (0.39) ALDH1A1TSHRPOLBGAAMAPT
SCHEMBL7050911 0.82 EPAS1 (0.34)
SCHEMBL7051891 0.81 ALDH1A1 (0.32) ALDH1A1POLBGAAMAPTMPI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0706396-B1 1,2,3,4-TETRAHYDROQUINOLINE-2,3,4-TRIONE-3 OR 4-OXIMES AND USE OREGON STATE (US) 2003-05-02 EP disclosed
US-5652368-A NERVOUS SYSTEM DISORDERS, ALZHEIMER'S DISEASE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-07-29 US disclosed
US-5475007-A Preventing convulsions THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-12-12 US disclosed