SCHEMBL7051912

SCHEMBL7051912

C[C@H]1CC[C@](c2cccc(NC(=O)c3cccc(F)c3)c2)(N2CCN(c3ccccc3)CC2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY1R P25929 2/20 0.52
MAPT P10636 4/20 0.52
TSHR P16473 2/20 0.52
LMNA P02545 2/20 0.52
KDM4E B2RXH2 2/20 0.52
NPSR1 Q6W5P4 1/20 0.52
NPC1 O15118 6/20 0.50
RAB9A P51151 6/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
TP53 P04637 2/20 0.50
KMT2A Q03164 6/20 0.48
MEN1 O00255 4/20 0.48
KCNK3 O14649 2/20 0.48
HPGD P15428 2/20 0.45
USP2 O75604 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
KCNK9 Q9NPC2 1/20 0.43
BTK Q06187 1/20 0.43
HTT P42858 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7051909 1.00 NPY1R (0.52) NPY1RMAPTTSHRLMNAKDM4E
SCHEMBL7055965 0.93 NPY1R (0.57) NPY1RMAPTTSHRKDM4ENPC1
SCHEMBL7055961 0.93 NPY1R (0.57) NPY1RMAPTTSHRKDM4ENPC1
SCHEMBL7049983 0.92 NPY1R (0.53) NPY1RMAPTTSHRLMNAKDM4E
SCHEMBL7049987 0.92 NPY1R (0.53) NPY1RMAPTTSHRLMNAKDM4E
SCHEMBL7057347 0.90 NPY1R (0.52) NPY1RMAPTTSHRLMNAKDM4E
SCHEMBL7057346 0.90 NPY1R (0.52) NPY1RMAPTTSHRLMNAKDM4E
SCHEMBL6992385 0.90 NPY1R (0.55) NPY1RMAPTTSHRLMNANPC1
SCHEMBL7054631 0.89 TDP1 (0.53) NPY1RMAPTLMNAKDM4ENPC1
SCHEMBL7054632 0.89 TDP1 (0.53) NPY1RMAPTLMNAKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6316617-B1 FOR TREATING PHYSIOLOGICAL DISORDERS ASSOCIATED WITH AN EXCESS OF NEUROPEPTIDE Y, SUCH AS FEEDING DISORDERS AND CERTAIN CARDIOVASCULAR DISEASES, MEDICAL DIAGNOSIS NEUROGEN CORPORATION 2001-11-13 US claimed
EP-0918761-B1 CERTAIN AMIDO- AND AMINO-SUBSTITUTED BENZYLAMINE DERIVATIVES; A NEW CLASS OF NEUROPEPTITE Y1 SPECIFIC LIGANDS NEUROGEN CORP (US) 2003-05-02 EP disclosed
US-6316617-B1 FOR TREATING PHYSIOLOGICAL DISORDERS ASSOCIATED WITH AN EXCESS OF NEUROPEPTIDE Y, SUCH AS FEEDING DISORDERS AND CERTAIN CARDIOVASCULAR DISEASES, MEDICAL DIAGNOSIS NEUROGEN CORPORATION 2001-11-13 US disclosed
US-6133265-A Certain amido- and amino- substituted benzylamine derivatives; a new class of neuropeptide Y1 specific ligands NEUROGEN CORPORATION (US) 2000-10-17 US disclosed