SCHEMBL7052182

SCHEMBL7052182

O=C1Nc2c(cc(Cl)c(Cl)c2[N+](=O)[O-])C(=O)/C1=N/O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.42
GRIN2D O15399 4/20 0.39
GRIN3B O60391 4/20 0.39
GRIN1 Q05586 4/20 0.39
GRIN2A Q12879 4/20 0.39
GRIN2B Q13224 4/20 0.39
GRIN2C Q14957 4/20 0.39
GRIN3A Q8TCU5 4/20 0.39
CES1 P23141 4/20 0.35
DNMT1 P26358 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.33
ALDH1A1 P00352 2/20 0.33
MAPT P10636 1/20 0.31
HSP90AA1 P07900 1/20 0.31
CDK5 Q00535 1/20 0.31
CDK5R1 Q15078 1/20 0.31
NCOA1 Q15788 1/20 0.31
NCOA3 Q9Y6Q9 1/20 0.31
GLP1R P43220 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7052184 1.00 TSHR (0.42) TSHRGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL7048389 0.90 TSHR (0.42) TSHRGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL7048387 0.90 TSHR (0.42) TSHRGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8872178 0.84 TSHR (0.52) TSHRGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL7054965 0.82 TSHR (0.36) TSHRGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL7052629 0.82 CES1 (0.41) CES1DNMT1SIRT2
SCHEMBL7052625 0.82 CES1 (0.41) CES1DNMT1SIRT2
SCHEMBL7050715 0.79 TSHR (0.42) TSHRGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL7050717 0.79 TSHR (0.42) TSHRGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL7053794 0.79 ALDH1A1 (0.33) ALDH1A1MAPTHSP90AA1CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0706396-B1 1,2,3,4-TETRAHYDROQUINOLINE-2,3,4-TRIONE-3 OR 4-OXIMES AND USE OREGON STATE (US) 2003-05-02 EP disclosed
US-5652368-A NERVOUS SYSTEM DISORDERS, ALZHEIMER'S DISEASE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-07-29 US disclosed
US-5475007-A Preventing convulsions THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-12-12 US disclosed