SCHEMBL7054978

SCHEMBL7054978

CC(=O)ON=C1C(=O)Nc2ccc(Br)c(C(F)(F)F)c2C1=O

nearest known ligand 0.32

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 2/20 0.32
AURKB Q96GD4 2/20 0.31
AURKC Q9UQB9 2/20 0.31
AURKA O14965 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31
CCNB2 O95067 1/20 0.31
CDK1 P06493 1/20 0.31
CCNB1 P14635 1/20 0.31
AHR P35869 1/20 0.31
GSK3A P49840 1/20 0.31
GSK3B P49841 1/20 0.31
CDK5 Q00535 1/20 0.31
CDK5R1 Q15078 1/20 0.31
CCNB3 Q8WWL7 1/20 0.31
TGM2 P21980 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7048384 0.91 AURKB (0.31) AGTR1AURKBAURKCAURKACCNB2
SCHEMBL7048274 0.87 GSK3A (0.31) AURKBAURKCAURKAGSK3AGSK3B
SCHEMBL7054468 0.86 CES1 (0.40) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL7048371 0.84 KMT2A (0.36) MEN1KMT2AALDH1A1MAPTHTT
SCHEMBL7052365 0.81 ALDH1A1 (0.32) AGTR1MEN1KMT2AALDH1A1MAPT
SCHEMBL7052368 0.81 ALDH1A1 (0.32) AGTR1MEN1KMT2AALDH1A1MAPT
SCHEMBL7051913 0.79 GALR3 (0.31) TGM2
SCHEMBL7054407 0.78 GSK3A (0.31) AURKBAURKCAURKAGSK3AGSK3B
SCHEMBL7053356 0.77 CES1 (0.43) ALDH1A1MAPTCCNB2CDK1CCNB1
SCHEMBL7055737 0.74 CES1 (0.38) CCNB2CDK1CCNB1GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0706396-B1 1,2,3,4-TETRAHYDROQUINOLINE-2,3,4-TRIONE-3 OR 4-OXIMES AND USE OREGON STATE (US) 2003-05-02 EP disclosed
US-5652368-A NERVOUS SYSTEM DISORDERS, ALZHEIMER'S DISEASE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-07-29 US disclosed
US-5475007-A Preventing convulsions THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-12-12 US disclosed