SCHEMBL7059534

SCHEMBL7059534

CNC(=O)Nc1sc(-c2ccccc2)cc1C(=O)NC(N)=O

nearest known ligand 0.73

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 7/20 0.73
MAP4K4 O95819 1/20 0.73
IKBKB O14920 3/20 0.60
JAK2 O60674 1/20 0.60
JAK3 P52333 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7051438 0.88 CHEK1 (0.82) CHEK1MAP4K4IKBKBJAK2JAK3
SCHEMBL7052328 0.88 CHEK1 (0.78) CHEK1MAP4K4IKBKBJAK2JAK3
SCHEMBL7055999 0.87 CHEK1 (0.72) CHEK1MAP4K4IKBKBJAK2JAK3
SCHEMBL5898667 0.87 IKBKB (0.74) CHEK1MAP4K4IKBKBJAK2JAK3
SCHEMBL7056909 0.86 IKBKB (0.82) CHEK1MAP4K4IKBKBJAK2JAK3
SCHEMBL7055226 0.84 CHEK1 (1.00) CHEK1MAP4K4IKBKBJAK2JAK3
SCHEMBL7055239 0.79 CHEK1 (1.00) CHEK1MAP4K4IKBKBJAK2JAK3
SCHEMBL7058336 0.79 CHEK1 (0.66) CHEK1MAP4K4IKBKBJAK2JAK3
SCHEMBL13930115 0.79 IKBKB (0.78) CHEK1MAP4K4IKBKBJAK2JAK3
SCHEMBL7055995 0.78 CHEK1 (0.62) CHEK1MAP4K4IKBKBJAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003029241-A1 CHK1 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-04-10 WO disclosed