SCHEMBL7060296

SCHEMBL7060296

c1cc(C2C[N]CCO2)ccn1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
TSHR P16473 1/20 0.30
MAPT P10636 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1515349 0.82 TSHR (0.50) CYP2C19TSHR
SCHEMBL5651938 0.82 TSHR (0.50) CYP2C19TSHR
SCHEMBL5651945 0.82 TSHR (0.50) CYP2C19TSHR
SCHEMBL5652143 0.79 MAOB (0.37)
SCHEMBL4968601 0.79 SLC6A2 (0.38)
SCHEMBL4971437 0.79 CYP3A4 (0.37) CYP1A2CYP2C19MAPT
SCHEMBL4968605 0.79 SLC6A2 (0.38)
SCHEMBL5654186 0.79 MAOB (0.37)
SCHEMBL4972142 0.79 MAOB (0.37)
SCHEMBL4971432 0.79 CYP3A4 (0.37) CYP1A2CYP2C19MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1309589-A2 UREA COMPOUNDS AND METHODS OF USES Amgen Inc. (US) 2003-05-14 EP disclosed
WO-2002014311-A2 UREA COMPOUNDS AND METHODS OF USES AMGEN INC. (US) 2002-02-21 WO disclosed
US-5773437-A UROGENITAL DISORDERS SUCH AS DYSURIA NIPPON CHEMIPHAR CO., LTD. (JP) 1998-06-30 US disclosed