SCHEMBL7063350

SCHEMBL7063350

COc1ccc(C(C)OC)cc1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.50
CA2 P00918 3/20 0.50
CA1 P00915 2/20 0.50
PPARG P37231 1/20 0.50
PPARD Q03181 1/20 0.50
PPARA Q07869 1/20 0.50
L3MBTL1 Q9Y468 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
KMT2A Q03164 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
CA12 O43570 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
MAPT P10636 3/20 0.46
CRHBP P24387 1/20 0.46
CRHR2 Q13324 1/20 0.46
PKM P14618 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13955907 0.84 PPARG (0.55) ACHECA2CA1PPARGPPARD
SCHEMBL12062531 0.83 SLC6A2 (0.43) ACHEMAPTCRHBPCRHR2PKM
SCHEMBL84033 0.82 PPARG (0.53) ACHECA2CA1PPARGPPARD
SCHEMBL30474606 0.82 TSHR (0.59) ACHEKMT2ANPSR1
SCHEMBL14515694 0.82 TSHR (0.59) ACHEKMT2ANPSR1
SCHEMBL21336451 0.82 GRM2 (0.43) ACHECA2CA1PPARGPPARD
SCHEMBL8859133 0.80 PPARG (0.52) ACHECA2CA1PPARGPPARD
SCHEMBL18553002 0.80 PPARG (0.52) ACHECA2CA1PPARGPPARD
SCHEMBL7430435 0.79 PPARG (0.51) ACHECA2CA1PPARGPPARD
SCHEMBL10343314 0.79 HIF1A (0.51) ACHECA2CA1PPARGPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000005-B1 PROCESS FOR THE PREPARATION OF 1-(3,4-DIMETHOXYPHENYL)ETHANOL AGRO CHEMIE NOEVENYVEDOESZER G (HU) 2003-05-21 EP disclosed
US-6403843-B1 REDUCTION OF 3,4-DIMETHOXYACETOPHENONE WITH HYDROGEN UNDER AQUEOUS CONDITIONS USING A RANEY NICKEL CATALYST; HIGH YIELD; PRODUCT CRYSTALS CAN BE EASILY FILTERED AGRO-CHEMIE (HU) 2002-06-11 US disclosed
EP-1000005-A1 PROCESS FOR THE PREPARATION OF 1-(3,4-DIMETHOXYPHENYL)ETHANOL Agro-Chemie Növenyvedöszer Gyárto Ertékesito Es Forgalmazo KFT. (HU) 2000-05-17 EP disclosed
WO-1999006343-A1 PROCESS FOR THE PREPARATION OF 1-(3,4-DIMETHOXYPHENYL)ETHANOL AGRO-CHEMIE NÖVENYVEDÖSZER GYARTO ERTEKESITÖ ES FORGALMAZO KFT. (HU) 1999-02-11 WO disclosed