SCHEMBL7068189

SCHEMBL7068189

CO[C@H](CC(=O)OC(C)(C)C)[C@H](C(C)C)N(C)C(=O)[C@@H](N)C(C)C

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.35
DPP4 P27487 2/20 0.33
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708027 0.90 CYP2D6 (0.33) CYP2D6DPP4
SCHEMBL13374875 0.90 CYP2D6 (0.33) CYP2D6DPP4
SCHEMBL25721685 0.90 CYP2D6 (0.33) CYP2D6DPP4
SCHEMBL17337592 0.90 CYP2D6 (0.33) CYP2D6DPP4
SCHEMBL17337593 0.90 CYP2D6 (0.33) CYP2D6DPP4
SCHEMBL18289855 0.90 CYP2D6 (0.33) CYP2D6DPP4
SCHEMBL14962705 0.90 CYP2D6 (0.33) CYP2D6DPP4
SCHEMBL21708028 0.90 CYP2D6 (0.33) CYP2D6DPP4
SCHEMBL18811712 0.83 CYP2D6 (0.33) CYP2D6DPP4
SCHEMBL18522915 0.82 CYP2D6 (0.32) CYP2D6DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0920325-A3 TETRAPEPTIDE DERIVATIVES OF DOLASTATIN AS ANTITUMOR AGENTS BASF AKTIENGESELLSCHAFT (DE) 2003-06-04 EP disclosed
EP-0920325-A2 TETRAPEPTIDE DERIVATIVES OF DOLASTATIN AS ANTITUMOR AGENTS BASF AKTIENGESELLSCHAFT (DE) 1999-06-09 EP disclosed
WO-1998004278-A2 TETRAPEPTIDE DERIVATIVES OF DOLASTATIN AS ANTITUMOR AGENTS BASF AKTIENGESELLSCHAFT (DE) 1998-02-05 WO disclosed